SCHEMBL6686504

SCHEMBL6686504

Cn1cccc1CNCCC[C@H](NC(=O)c1ccc(CNCc2cc[nH]n2)cc1)C(=O)O.NCc1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.41
FOLH1 Q04609 4/20 0.39
CASR P41180 1/20 0.36
FPGS Q05932 4/20 0.35
TGM2 P21980 1/20 0.34
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34
TPSAB1 Q15661 1/20 0.34
DHFR P00374 3/20 0.34
TYMS P04818 1/20 0.34
FNTA P49354 2/20 0.33
FNTB P49356 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
PGGT1B P53609 1/20 0.33
KLKB1 P03952 1/20 0.33
C3AR1 Q16581 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6018574 0.89 CXCR4 (0.51) CXCR4FOLH1CASRTGM2PRSS1
SCHEMBL6017964 0.89 CXCR4 (0.43) CXCR4FOLH1PRSS1PRSS2PRSS3
SCHEMBL6687483 0.88 CXCR4 (0.40) CXCR4FOLH1CASRFPGSTGM2
SCHEMBL6682711 0.86 CXCR4 (0.40) CXCR4FOLH1CASRFPGSTGM2
SCHEMBL6690573 0.85 HDAC1 (0.40) CXCR4FOLH1CASRFPGSDHFR
SCHEMBL6687885 0.84 FOLH1 (0.41) FOLH1CASRTGM2PRSS1PRSS2
SCHEMBL6681620 0.82 FOLH1 (0.43) FOLH1CASRTGM2DHFRC3AR1
SCHEMBL6689563 0.81 FOLH1 (0.45) CXCR4FOLH1CASRFPGSTGM2
SCHEMBL6018262 0.80 CXCR4 (0.57) CXCR4FOLH1CASRFPGSTGM2
SCHEMBL6018284 0.80 HDAC3 (0.47) CXCR4FOLH1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed