SCHEMBL6681620

SCHEMBL6681620

Cn1cccc1CNCCCC(NC(=O)c1ccc(C(N)Cc2cccn2C)cc1)C(=O)O.NCc1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 3/20 0.43
CASR P41180 2/20 0.39
C3AR1 Q16581 1/20 0.36
CCKBR P32239 1/20 0.35
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
TGM2 P21980 4/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CA2 P00918 2/20 0.33
MME P08473 1/20 0.33
ACE P12821 1/20 0.33
CPA1 P15085 1/20 0.33
ACE2 Q9BYF1 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681809 0.92 FOLH1 (0.39) FOLH1CASRC3AR1CCKBRITGB3
SCHEMBL6685296 0.90 FOLH1 (0.38) FOLH1CASRC3AR1CCKBRITGB3
SCHEMBL6688643 0.90 FOLH1 (0.38) FOLH1CASRC3AR1CCKBRHTT
SCHEMBL6683363 0.85 FOLH1 (0.41) FOLH1CASRC3AR1CCKBRITGB3
SCHEMBL6687885 0.83 FOLH1 (0.41) FOLH1CASRTGM2CYP3A4
SCHEMBL6682711 0.83 CXCR4 (0.40) FOLH1CASRTGM2HTTSMN1; SMN2
SCHEMBL6018574 0.83 CXCR4 (0.51) FOLH1CASRTGM2DHFR
SCHEMBL6687483 0.82 CXCR4 (0.40) FOLH1CASRTGM2DHFR
SCHEMBL6686504 0.82 CXCR4 (0.41) FOLH1CASRC3AR1TGM2DHFR
SCHEMBL6690573 0.81 HDAC1 (0.40) FOLH1CASRDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed