SCHEMBL6687347

SCHEMBL6687347

COc1ccc(-n2nc(OCC3CCCCC3)nc2-c2ccc(O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.56
PTGS2 P35354 4/20 0.56
MALT1 Q9UDY8 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.40
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CCNA1 P78396 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
CNR1 P21554 3/20 0.40
CNR2 P34972 3/20 0.40
MGLL Q99685 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ESR1 P03372 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687157 0.99 PTGS1 (0.57) PTGS1PTGS2MALT1L3MBTL1CCNB2
SCHEMBL6687131 0.95 PTGS1 (0.60) PTGS1PTGS2MALT1L3MBTL1MGLL
SCHEMBL6687111 0.87 PTGS1 (0.52) PTGS1PTGS2MALT1L3MBTL1MGLL
SCHEMBL6687447 0.84 PTGS1 (0.57) PTGS1PTGS2MALT1L3MBTL1MAPT
SCHEMBL6681046 0.84 PTGS2 (0.60) PTGS1PTGS2MALT1L3MBTL1CNR1
SCHEMBL6686621 0.82 PTGS1 (0.54) PTGS1PTGS2MALT1L3MBTL1MGLL
SCHEMBL6683372 0.79 PTGS1 (0.69) PTGS1PTGS2MALT1L3MBTL1ESR2
SCHEMBL6682126 0.78 MALT1 (0.53) PTGS1PTGS2MALT1L3MBTL1
SCHEMBL6132456 0.78 PTGS2 (0.67) PTGS1PTGS2MALT1L3MBTL1CNR1
SCHEMBL6684493 0.78 PTGS1 (0.60) PTGS1PTGS2MALT1L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060367-A1 IMIDAZOLE AND TRIAZOLE DERIVATIVES USEFUL AS SELECTIVE COX-1 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-22 WO disclosed