SCHEMBL6688684

SCHEMBL6688684

N#Cc1ccc2c(c1)S(=O)(=O)N=C(c1c(O)c3cc(F)ccc3n(CCC3CC3)c1=O)N2

nearest known ligand 0.78

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.78
NR1I2 O75469 1/20 0.78
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PLK1 P53350 5/20 0.38
L3MBTL1 Q9Y468 1/20 0.34
DRD2 P14416 3/20 0.33
DRD3 P35462 3/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
HTR1D P28221 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
PADI4 Q9UM07 1/20 0.32
CRY1 Q16526 1/20 0.32
CRY2 Q49AN0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690316 0.90 CYP2C9 (0.83) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6693468 0.90 CYP2C9 (0.81) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6232054 0.89 CYP2C9 (0.80) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6234934 0.88 CYP2C9 (0.79) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL5089690 0.88 CYP2C9 (1.00) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6689772 0.87 CYP2C9 (0.78) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6687473 0.87 CYP2C9 (0.77) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6236224 0.87 CYP2C9 (0.80) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6693467 0.86 CYP2C9 (0.79) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6689094 0.86 CYP2C9 (0.76) CYP2C9NR1I2MAPK1HSD17B10PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO disclosed