SCHEMBL6690285

SCHEMBL6690285

COc1cc(CNC(Cc2ccccc2)C(N)=O)ccc1OCc1c(F)cccc1F

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
PKM P14618 1/20 0.47
CTSD P07339 6/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
MRGPRX1 Q96LB2 2/20 0.46
HTT P42858 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
F2 P00734 1/20 0.46
F10 P00742 1/20 0.46
PRSS1 P07477 1/20 0.46
F7 P08709 1/20 0.46
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6685320 1.00 KMT2A (0.55) KMT2AMEN1CYP3A4CYP2C19RAB9A
SCHEMBL6690750 0.94 KMT2A (0.53) KMT2AMEN1CYP3A4CYP2C19RAB9A
SCHEMBL6690744 0.94 KMT2A (0.53) KMT2AMEN1CYP3A4CYP2C19RAB9A
SCHEMBL6686902 0.89 NPC1 (0.58) KMT2AMEN1RAB9ANPC1PKM
SCHEMBL6686899 0.89 NPC1 (0.58) KMT2AMEN1RAB9ANPC1PKM
SCHEMBL6690108 0.88 SMN1; SMN2 (0.56) KMT2AMEN1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL6690105 0.88 SMN1; SMN2 (0.56) KMT2AMEN1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL6686469 0.87 KMT2A (0.53) KMT2AMEN1RAB9ANPC1PKM
SCHEMBL6686470 0.87 KMT2A (0.53) KMT2AMEN1RAB9ANPC1PKM
SCHEMBL6687911 0.86 KMT2A (0.56) KMT2AMEN1SMN1; SMN2HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed