SCHEMBL6690764

SCHEMBL6690764

CC(C)CC(NCc1ccc(OCc2c(F)cccc2Cl)c([N+](=O)[O-])c1)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 11/20 0.46
CD274 Q9NZQ7 11/20 0.46
SMN1; SMN2 Q16637 1/20 0.42
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.38
S1PR1 P21453 1/20 0.38
S1PR5 Q9H228 1/20 0.38
DHODH Q02127 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6689254 0.83 SCN9A (0.53)
SCHEMBL6689256 0.83 SCN9A (0.53)
SCHEMBL6686767 0.82 CD274 (0.53) PDCD1CD274SMN1; SMN2KMT2AMEN1
SCHEMBL6686469 0.79 KMT2A (0.53) SMN1; SMN2KMT2AMEN1GAARAB9A
SCHEMBL6686470 0.79 KMT2A (0.53) SMN1; SMN2KMT2AMEN1GAARAB9A
SCHEMBL6688731 0.78 CD274 (0.45) PDCD1CD274SMN1; SMN2KMT2AMEN1
SCHEMBL6688726 0.78 CD274 (0.45) PDCD1CD274SMN1; SMN2KMT2AMEN1
SCHEMBL6254681 0.78 PDCD1 (0.41) PDCD1CD274SMN1; SMN2KMT2AMEN1
SCHEMBL6254676 0.78 PDCD1 (0.41) PDCD1CD274SMN1; SMN2KMT2AMEN1
SCHEMBL6694008 0.78 PDCD1 (0.44) PDCD1CD274RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed