SCHEMBL6694982

SCHEMBL6694982

Cc1cc(I)ccc1Nc1ccccc1C(=O)NCCO

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 6/20 0.53
MAP2K2 P36507 3/20 0.53
IDO1 P14902 1/20 0.44
PTGS2 P35354 6/20 0.44
GPR52 Q9Y2T5 1/20 0.43
MT-CO2 P00403 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
PTGS1 P23219 2/20 0.43
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6035241 0.91 MAP2K1 (0.53) MAP2K1MAP2K2IDO1KDM4EALDH1A1
SCHEMBL6035385 0.85 MAP2K1 (0.53) MAP2K1MAP2K2IDO1GPR52MT-CO2
SCHEMBL6035378 0.85 MAP2K1 (0.48) MAP2K1MAP2K2IDO1KDM4EALDH1A1
SCHEMBL5676551 0.85 HPGD (0.55) MAP2K1MAP2K2IDO1GPR52
SCHEMBL6035461 0.84 MAP2K1 (0.55) MAP2K1MAP2K2IDO1GPR52JAK1
SCHEMBL6036120 0.84 KMT2A (0.49) MAP2K1MAP2K2KDM4EALDH1A1MAPT
SCHEMBL27583296 0.82 MAP2K1 (0.61) MAP2K1MAP2K2PTGS2GPR52JAK1
SCHEMBL15603461 0.82 MAP2K1 (0.70) MAP2K1MAP2K2
SCHEMBL7715685 0.82 IDO1 (0.48) MAP2K1MAP2K2IDO1PTGS2KDM4E
SCHEMBL6036200 0.82 KMT2A (0.48) MAP2K1MAP2K2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696440-B1 ADMINISTERING MITOGEN ACTIVATED PROTEIN KINASE(MEK) INHIBITORS COMPRISING SECONDARY CARBOCYCLIC AMINES, AS ANTIASTHMATIC AGENTS WARNER-LAMBERT COMPANY 2004-02-24 US disclosed