SCHEMBL6695038

SCHEMBL6695038

NCC1(c2ccccc2)CCN(CCC(c2ccccc2)(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.53
MAOB P27338 1/20 0.53
TAAR1 Q96RJ0 1/20 0.53
DPP4 P27487 2/20 0.50
CCR1 P32246 3/20 0.48
KCNA3 P22001 2/20 0.46
CCR3 P51677 1/20 0.44
OPRM1 P35372 3/20 0.43
LMNA P02545 1/20 0.43
CHRM2 P08172 1/20 0.43
HTR1A P08908 1/20 0.43
CYP2D6 P10635 1/20 0.43
CHRM1 P11229 1/20 0.43
KCNH2 Q12809 1/20 0.43
SLC6A4 P31645 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KIF11 P52732 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11603149 0.99 MAOA (0.51) MAOAMAOBTAAR1DPP4CCR1
Hydrochloric Acid SCHEMBL11602646 0.99 MAOA (0.51) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11656657 0.92 MAOA (0.45) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11602768 0.92 MAOA (0.45) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11602929 0.92 MAOA (0.45) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11601863 0.92 CCR1 (0.53) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11603862 0.92 CCR1 (0.53) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11601401 0.92 MEN1 (0.49) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11601959 0.92 MEN1 (0.49) MAOAMAOBTAAR1DPP4CCR1
SCHEMBL11602881 0.91 CCR1 (0.51) MAOAMAOBTAAR1DPP4CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3553083-B2 2004-08-11 JP claimed
EP-0852494-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-07-15 EP claimed
WO-1997009973-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-03-20 WO claimed
US-4069223-A ANTIDIARRHEA G. D. SEARLE & CO. (US) 1978-01-17 US claimed
US-6576650-B1 No central nervous system side effects REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-06-10 US disclosed
US-6573282-B1 Compositions for treatment of peripheral hyperalgesia are provided. The compositions contain an anti-hyperalgesia effective amount of one or more compounds that directly or indirectly interact with peripheral opiate receptors ADOLOR CORPORATION 2003-06-03 US disclosed
US-6166039-A Peripherally active anti-hyperalgesic opiates REGENTS OF THE UNIV. OF CALIFORNIA (US) 2000-12-26 US disclosed
US-5994372-A ANTIDIARRHEA COMPOUND REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-11-30 US disclosed
US-5849761-A Peripherally active anti-hyperalgesic opiates REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-12-15 US disclosed
US-4069223-A ANTIDIARRHEA G. D. SEARLE & CO. (US) 1978-01-17 US disclosed