SCHEMBL6695693

SCHEMBL6695693

c1ccc(Cc2ccccc2[C](c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.55
CYP2D6 P10635 3/20 0.50
CYP2C19 P33261 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 2/20 0.50
BCL2 P10415 1/20 0.47
BCL2L1 Q07817 1/20 0.47
CYP3A4 P08684 2/20 0.45
CALM1 P0DP23 1/20 0.44
HTR2A P28223 1/20 0.44
CAPN1 P07384 1/20 0.43
PTPN1 P18031 1/20 0.41
ALOX5 P09917 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
NFKB1 P19838 1/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6272312 0.82 TSHR (0.62) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL9806310 0.82 TSHR (0.53) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL28259941 0.82 TSHR (0.53) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
Thiobenzoic Acid SCHEMBL7714480 0.79 TSHR (0.50) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
Benzoic Acid SCHEMBL29974267 0.79 TSHR (0.86) TSHRCAPN1PTPN1CA1CA2
SCHEMBL1046696 0.79 TSHR (0.59) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL5597331 0.77 TSHR (0.52) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL23003 0.77 TSHR (0.79) TSHRCYP2C9CAPN1PTPN1CA1
SCHEMBL1247034 0.77 TSHR (0.61) TSHRCYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL9365256 0.77 TSHR (0.52) TSHRCYP2D6CYP2C19CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040171881-A1 N,N'-substituted-1,3-diamino-2-hydroxypropane derivatives PHARMACIA & UPJOHN COMPANY 2004-09-02 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040171881-A1 N,N'-substituted-1,3-diamino-2-hydroxypropane derivatives BACE1, BACE2, PSEN1 TSHR 3190/4885CYP2D6 2162/4885CYP2C19 3144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.