SCHEMBL6697523

SCHEMBL6697523

NC(Cn1ccnc1)c1ccccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.53
IDO1 P14902 3/20 0.49
ADRA2C P18825 1/20 0.48
ALOX15 P16050 3/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP3A4 P08684 4/20 0.46
CYP1A2 P05177 3/20 0.46
CYP2D6 P10635 3/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
TBXAS1 P24557 1/20 0.46
QPCT Q16769 1/20 0.46
CYP4Z1 Q86W10 1/20 0.46
QPCTL Q9NXS2 1/20 0.46
TSHR P16473 3/20 0.45
CYP2C9 P11712 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6312314 0.88 CYP3A4 (0.46) CYP19A1IDO1ADRA2CALOX15ALDH1A1
SCHEMBL9367826 0.86 CYP19A1 (0.57) CYP19A1IDO1ADRA2CALOX15ALDH1A1
SCHEMBL31180917 0.82 ADRA2C (0.71) CYP19A1IDO1ADRA2CALOX15CYP3A4
SCHEMBL6313011 0.82 ADRA2C (0.59) CYP19A1IDO1ADRA2CALOX15CYP3A4
SCHEMBL6305279 0.82 ADRA2C (0.71) CYP19A1IDO1ADRA2CALOX15CYP3A4
SCHEMBL6305674 0.82 ADRA2C (0.71) CYP19A1IDO1ADRA2CALOX15CYP3A4
SCHEMBL29669977 0.82 ADRA2C (0.70) CYP19A1IDO1ADRA2CAGER
SCHEMBL11277181 0.82 ADRA2C (0.70) CYP19A1IDO1ADRA2CAGER
SCHEMBL6394302 0.80 ADRA2C (0.44) CYP19A1IDO1ADRA2CALOX15CYP3A4
SCHEMBL3670452 0.78 CYP19A1 (0.58) CYP19A1CYP3A4CYP1A2CYP2D6POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040039033-A1 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial F1F0 ATP hydrolase BRISTOL-MYERS SQUIBB COMPANY 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039033-A1 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial F1F0 ATP hydrolase ATP5F1A, ATP5ME, ATP5F1D CYP19A1 3335/4885IDO1 3414/4885ADRA2C 783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.