SCHEMBL6698196

SCHEMBL6698196

CCC1=CC(=O)C2(Cc3ccccc3)CN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CCN12

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 17/20 0.59
UGCG Q16739 2/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6698193 1.00 GHSR (0.59) GHSRUGCGCYP3A4
SCHEMBL6694789 0.91 GHSR (0.59) GHSRUGCGCYP3A4
SCHEMBL6698203 0.85 GHSR (0.53) GHSRUGCGCYP3A4
SCHEMBL6689376 0.85 GHSR (0.53) GHSRUGCGCYP3A4
SCHEMBL6698202 0.85 GHSR (0.53) GHSRUGCGCYP3A4
SCHEMBL5228711 0.85 GHSR (0.64) GHSRUGCGCYP3A4
SCHEMBL5226702 0.85 GHSR (0.64) GHSRUGCGCYP3A4
SCHEMBL6691393 0.85 GHSR (0.53) GHSRUGCGCYP3A4
SCHEMBL6691993 0.85 GHSR (0.53) GHSRUGCGCYP3A4
SCHEMBL6691397 0.85 GHSR (0.53) GHSRUGCGCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1002802-B1 Dipeptide derivatives as growth hormone secretagogues PFIZER PROD INC (US) 2004-12-08 EP claimed
US-6194578-B1 GROWTH HORMONE SECRETAGOGUES; USEFUL FOR PROPHYLAXIS AND THERAPY OF OSTEOPOROSIS AND/OR FRAILTY, INSULIN RESISTANCE IN MAMMALS, CONGESTIVE HEART FAILURE, OBESITY, ACCELERATING BONE FRACTURE REPAIR REDUCING CACHEXIA AND PROTEIN LOSS PFIZER INC. 2001-02-27 US claimed
EP-1002802-A1 Dipeptide derivatives as growth hormone secretagogues Pfizer Products Inc. (US) 2000-05-24 EP claimed
EP-1002802-B1 Dipeptide derivatives as growth hormone secretagogues PFIZER PROD INC (US) 2004-12-08 EP disclosed
US-6194578-B1 GROWTH HORMONE SECRETAGOGUES; USEFUL FOR PROPHYLAXIS AND THERAPY OF OSTEOPOROSIS AND/OR FRAILTY, INSULIN RESISTANCE IN MAMMALS, CONGESTIVE HEART FAILURE, OBESITY, ACCELERATING BONE FRACTURE REPAIR REDUCING CACHEXIA AND PROTEIN LOSS PFIZER INC. 2001-02-27 US disclosed
EP-1002802-A1 Dipeptide derivatives as growth hormone secretagogues Pfizer Products Inc. (US) 2000-05-24 EP disclosed