SCHEMBL6700628

SCHEMBL6700628

Cn1nccc1Nc1nc(-c2ccc(-c3ccccc3)cc2)nc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 9/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
PDE5A O76074 7/20 0.55
TGFBR1 P36897 1/20 0.54
MAPK14 Q16539 1/20 0.54
KDM1A O60341 2/20 0.54
LMNA P02545 2/20 0.53
MAPT P10636 2/20 0.53
TP53 P04637 1/20 0.53
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
POLB P06746 1/20 0.51
HPGD P15428 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7123370 0.91 ABCG2 (0.60) ABCG2MEN1KMT2APDE5ATGFBR1
SCHEMBL7155962 0.86 ABCG2 (0.59) ABCG2MEN1KMT2APDE5ATGFBR1
SCHEMBL1798811 0.81 PDE5A (0.54) ABCG2MEN1KMT2APDE5ATGFBR1
SCHEMBL7234183 0.77 MEN1 (0.51) ABCG2MEN1KMT2APDE5ATGFBR1
SCHEMBL4856833 0.73 PDE5A (0.64) MEN1KMT2APDE5ALMNATP53
SCHEMBL7124846 0.73 NPY5R (0.57) KDM1ATP53SMN1; SMN2
SCHEMBL1063103 0.73 ABCG2 (1.00) ABCG2MEN1KMT2APDE5ATGFBR1
SCHEMBL14474836 0.72 ABCG2 (0.62) ABCG2MEN1KMT2ALMNAMAPT
SCHEMBL1063009 0.72 ABCG2 (0.69) ABCG2MEN1KMT2APDE5ATGFBR1
SCHEMBL5675207 0.71 ABCG2 (0.61) ABCG2MEN1KMT2AGSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116454-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2004-06-17 US disclosed