SCHEMBL670630

SCHEMBL670630

CC(C)(C)c1nc(CN(C(=O)O)C(C)(C)C)n(-c2cccc(Cl)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 10/20 0.40
PKM P14618 1/20 0.40
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
GRM5 P41594 2/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PPP1CA P62136 1/20 0.37
SLC16A3 O15427 2/20 0.37
SLC16A1 P53985 2/20 0.37
MCTS1 Q9ULC4 1/20 0.37
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12506473 0.81 TRPV1 (0.49) TRPV1PKMHDAC1HDAC6
SCHEMBL10093696 0.78 TRPV1 (0.41) TRPV1PKMALDH1A1LMNAGAA
Hydrochloric Acid SCHEMBL656099 0.77 TRPV1 (0.40) TRPV1PKMALDH1A1LMNAGAA
SCHEMBL12506475 0.77 PKM (0.43) TRPV1PKMALDH1A1KDM4ELMNA
SCHEMBL10186767 0.75 TRPV1 (0.46) TRPV1HDAC1HDAC6
SCHEMBL10093694 0.72 TRPV1 (0.44) TRPV1HDAC1HDAC6
SCHEMBL287641 0.70 TRPV1 (0.66) TRPV1
SCHEMBL288083 0.69 TRPV1 (0.71) TRPV1
SCHEMBL2688133 0.68 MAPK14 (0.51) TRPV1PKM
SCHEMBL287373 0.68 TRPV1 (0.56) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606033-A1 SUBSTITUTED CYCLIC CARBOXAMIDE AND UREA DERIVATIVES AS LIGANDS OF THE VANILLOID RECEPTOR Grünenthal GmbH (DE) 2013-06-26 EP disclosed
WO-2012022487-A1 SUBSTITUTED CYCLIC CARBOXAMIDE AND UREA DERIVATIVES AS LIGANDS OF THE VANILLOID RECEPTOR Grünenthal GmbH (DE) 2012-02-23 WO disclosed