SCHEMBL6709246

SCHEMBL6709246

Cc1cc(N2CCCC2)c2ccc(NCCc3ccc(Cl)cc3)cc2n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.47
NCF1 P14598 3/20 0.47
MAPK1 P28482 3/20 0.42
LMNA P02545 2/20 0.42
USP2 O75604 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP3A4 P08684 3/20 0.41
CTNNB1 P35222 1/20 0.41
TCF7L2 Q9NQB0 1/20 0.41
CNR1 P21554 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5026871 0.89 NPC1 (0.52) NCF1MAPK1LMNAUSP2TSHR
SCHEMBL5028660 0.83 NCF1 (0.51) NCF1MAPK1LMNAUSP2TSHR
SCHEMBL5024388 0.81 CTNNB1 (0.49) NCF1CTNNB1TCF7L2
SCHEMBL5022706 0.80 NCF1 (0.51) NCF1
SCHEMBL5024554 0.80 NCF1 (0.51) NCF1HTTSMN1; SMN2CTNNB1TCF7L2
SCHEMBL5026876 0.78 NCF1 (0.46) NCF1CTNNB1TCF7L2
SCHEMBL5022553 0.78 NCF1 (0.51) NCF1MAPK1HTTCTNNB1TCF7L2
SCHEMBL5025329 0.78 NCF1 (0.53) NCF1MAPK1
SCHEMBL5024412 0.78 NCF1 (0.53) NCF1MAPK1LMNAUSP2HTT
SCHEMBL5026894 0.77 NCF1 (0.48) NCF1MAPK1LMNAUSP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474145-A1 QUINOLINE DERIVATIVES AS NPY ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-11-10 EP disclosed
WO-2003066055-A1 QUINOLINE DERIVATIVES AS NPY ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2003-08-14 WO disclosed