SCHEMBL6719741

SCHEMBL6719741

COc1cc(C(=O)CF)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.50
TSHR P16473 2/20 0.46
CTNNB1 P35222 2/20 0.46
WNT3A P56704 2/20 0.46
MAPT P10636 2/20 0.46
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA7 P43166 1/20 0.43
TPMT P51580 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13545220 0.85 MEN1 (0.59) PDE4DTSHRCTNNB1WNT3AMAPT
SCHEMBL8680313 0.84 TSHR (0.63) PDE4DTSHRCTNNB1WNT3AMAPT
SCHEMBL23112630 0.83 GSK3B (0.54) PDE4DTSHRCTNNB1WNT3AMAPT
SCHEMBL7482554 0.83 PDE4B (0.42) PDE4D
SCHEMBL6361805 0.82 PDE4D (0.49) PDE4DTSHRCTNNB1WNT3AMAPT
SCHEMBL16954378 0.81 MAPT (0.43) PDE4DTSHRMAPTLMNACYP1A2
SCHEMBL141068 0.81 HTT (0.49) TSHRCTNNB1WNT3AMAPTLMNA
SCHEMBL27456578 0.80 CYP1A2 (0.68) TSHRMAPTLMNACYP1A2CYP3A4
SCHEMBL7432445 0.80 MAPT (0.57) PDE4DTSHRCTNNB1WNT3AMAPT
SCHEMBL3856127 0.79 CYP1A2 (0.50) PDE4DTSHRMAPTLMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101270117-B Herbicide and preparation thereof UNIV DALIAN TECH 2012-02-29 CN claimed
CN-101279972-B Benzoxazole herbicides and preparation thereof UNIV DALIAN TECH 2011-02-02 CN claimed
CN-101870677-A 5-arylmethoxy phenyl pyrazole compound and preparation method thereof UNIV DALIAN TECH 2010-10-27 CN claimed
CN-101279972-A Benzoxazole herbicides and preparation thereof UNIV DALIAN TECH (CN) 2008-10-08 CN claimed
CN-101270117-A Herbicide and preparation thereof UNIV DALIAN TECH (CN) 2008-09-24 CN claimed
CN-101270117-B Herbicide and preparation thereof UNIV DALIAN TECH 2012-02-29 CN disclosed
CN-101279972-B Benzoxazole herbicides and preparation thereof UNIV DALIAN TECH 2011-02-02 CN disclosed
CN-101870677-A 5-arylmethoxy phenyl pyrazole compound and preparation method thereof UNIV DALIAN TECH 2010-10-27 CN disclosed
CN-101279972-A Benzoxazole herbicides and preparation thereof UNIV DALIAN TECH (CN) 2008-10-08 CN disclosed
CN-101270117-A Herbicide and preparation thereof UNIV DALIAN TECH (CN) 2008-09-24 CN disclosed
EP-0791571-B1 Benzoyl derivatives BAYER CROPSCIENCE AG (DE) 2004-06-16 EP disclosed
US-20040092402-A1 Pyrimidine derivatives and herbicides containing the same SUMITOMO CHEMICAL TAKEDA AGRO COMPANY, LIMITED (JP) 2004-05-13 US disclosed
CN-1090845-A Process for preparing substituted aryl-halogenoalkyl pyrazoles MONSANTO CO (US) 1994-08-17 CN disclosed
US-5281571-A Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles MONSANTO COMPANY (US) 1994-01-25 US disclosed
EP-0553307-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1993-08-04 EP disclosed
EP-0542872-A1 HERBICIDAL SUBSTITUTED ARYL ALKYLSULFONYL PYRAZOLES MONSANTO COMPANY (US) 1993-05-26 EP disclosed
CN-1061777-A Substituted aryl-haloalkyl-pyrazoles as herbicides MONSANTO CO (US) 1992-06-10 CN disclosed
CN-1061221-A The aryl alkylsulfonyl pyrazoles of the replacement of weeding MONSANTO CO (US) 1992-05-20 CN disclosed
WO-1992006962-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1992-04-30 WO disclosed
WO-1992002509-A1 HERBICIDAL SUBSTITUTED ARYL ALKYLSULFONYL PYRAZOLES MONSANTO COMPANY (US) 1992-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092402-A1 Pyrimidine derivatives and herbicides containing the same DDX41, CBR3, DPYD PDE4D 3003/4885TSHR 2182/4885CTNNB1 1654/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.