SCHEMBL8680313

SCHEMBL8680313

COc1ccc(C(=O)CF)cc1OC

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2C9 P11712 1/20 0.63
CYP2C19 P33261 1/20 0.63
MAPT P10636 5/20 0.63
CTNNB1 P35222 2/20 0.63
WNT3A P56704 2/20 0.63
CA12 O43570 1/20 0.61
CA1 P00915 1/20 0.61
CA2 P00918 1/20 0.61
CA4 P22748 1/20 0.61
CA6 P23280 1/20 0.61
CA7 P43166 1/20 0.61
TPMT P51580 1/20 0.61
CA9 Q16790 1/20 0.61
CA14 Q9ULX7 1/20 0.61
ALDH1A1 P00352 4/20 0.58
GAA P10253 2/20 0.55
MEN1 O00255 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18652086 0.89 MAPK1 (0.63) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL141068 0.86 HTT (0.49) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2848243 0.86 HTT (0.67) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10830384 0.86 PDE4B (0.57) TSHRMAPTCTNNB1WNT3AALDH1A1
SCHEMBL1659363 0.85 MAPT (0.71) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10455919 0.85 CTNNB1 (0.83) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6719741 0.84 PDE4D (0.50) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3893527 0.83 TSHR (0.66) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL29578705 0.83 MEN1 (0.73) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL515746 0.83 MEN1 (0.73) TSHRCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114873-B1 N-[3-BROMO-4-(3- [18F]FLUOROPROPOXY)-BENZYL]-GUANIDINE FOR IMAGING CARDIAC INNERVATION LANTHEUS MEDICAL IMAGING INC (US) 2013-02-20 EP disclosed
EP-2474526-A2 Ligands for imaging cardiac innervation Lantheus Medical Imaging, Inc. (US) 2012-07-11 EP disclosed
EP-2474525-A2 Ligands for imaging cardiac innervation Lantheus Medical Imaging, Inc. (US) 2012-07-11 EP disclosed
EP-2474523-A2 Ligands for imaging cardiac innervation Lantheus Medical Imaging, Inc. (US) 2012-07-11 EP disclosed
EP-2474524-A2 Ligands for imaging cardiac innervation Lantheus Medical Imaging, Inc. (US) 2012-07-11 EP disclosed
WO-2008083056-A2 LIGANDS FOR IMAGING CARDIAC INNERVATION LANTHEUS MEDICAL IMAGING, INC. (US) 2008-07-10 WO disclosed
WO-1998024740-A1 FLUORINATION OF CARBONYL-SUBSTITUTED AROMATIC COMPOUNDS F2 CHEMICALS LIMITED (GB) 1998-06-11 WO disclosed