SCHEMBL6722652

SCHEMBL6722652

CCOCc1cc(OCC)c(-c2ccc(C[C@H](NC(=O)c3c(F)cccc3F)C(=O)O)cc2)c(OCC)c1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 15/20 0.54
ITGB1 P05556 14/20 0.54
ITGB7 P26010 11/20 0.54
ITGB2 P05107 2/20 0.44
ICAM1 P05362 2/20 0.44
ITGAL P20701 2/20 0.44
ITGB3 P05106 1/20 0.44
ITGAV P06756 1/20 0.44
ALB P02768 1/20 0.43
IL2 P60568 1/20 0.43
KIFC1 Q9BW19 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Firategrast SCHEMBL918399 0.93 ITGA4 (0.54) ITGA4ITGB1ITGB7ALBIL2
Firategrast SCHEMBL12002530 0.93 ITGA4 (0.54) ITGA4ITGB1ITGB7ALBIL2
Firategrast SCHEMBL1681763 0.91 ITGA4 (0.53) ITGA4ITGB1ITGB7ALBIL2
SCHEMBL27499526 0.87 ITGA4 (0.56) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL919212 0.87 ITGA4 (0.56) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL12943224 0.87 ITGA4 (0.51) ITGA4ITGB1ITGB7ITGB2ICAM1
SCHEMBL919328 0.85 ITGA4 (0.53) ITGA4ITGB1ITGB7ALBIL2
SCHEMBL920095 0.85 ITGA4 (0.46) ITGA4ITGB1ITGB7
SCHEMBL920937 0.84 ITGA4 (0.47) ITGA4ITGB1ITGB7
SCHEMBL920085 0.84 ITGA4 (0.57) ITGA4ITGB1ITGB7ALBIL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478619-A1 A PROCESS FOR PREPARING A PHENYLALANINE DERIVATIVE AND INTERMEDIATES THEREOF TANABE SEIYAKU CO., LTD. (JP) 2004-11-24 EP disclosed
WO-2003072536-A1 A PROCESS FOR PREPARING A PHENYLALANINE DERIVATIVE AND INTERMEDIATES THEREOF TANABE SEIYAKU CO., LTD. (JP) 2003-09-04 WO disclosed