SCHEMBL673307

SCHEMBL673307

COC(=O)c1csc(Br)c1Br

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.59
CHEK1 O14757 1/20 0.42
MET P08581 1/20 0.42
GSK3B P49841 1/20 0.42
LIMK1 P53667 1/20 0.42
DYRK1A Q13627 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
GAA P10253 2/20 0.42
POLB P06746 2/20 0.42
LMNA P02545 1/20 0.38
HSD17B10 Q99714 3/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38
SLC6A3 Q01959 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15472134 0.82 KMT2A (0.44) TSHRCHEK1METGSK3BLIMK1
SCHEMBL16212689 0.82 TSHR (0.42) TSHRCHEK1METGSK3BLIMK1
SCHEMBL18490206 0.81 CHEK1 (0.41) TSHRCHEK1METGSK3BLIMK1
SCHEMBL29137861 0.79 TSHR (0.53) TSHRNPC1RAB9AGAAPOLB
SCHEMBL20263513 0.78 TSHR (0.39) TSHRCHEK1METGSK3BLIMK1
SCHEMBL1527614 0.75 CHEK1 (0.37) TSHRCHEK1METGSK3BLIMK1
SCHEMBL24716081 0.74 KMT2A (0.47) TSHRNPC1RAB9AGAAPOLB
SCHEMBL20607510 0.74 CHEK1 (0.47) TSHRCHEK1METGSK3BLIMK1
SCHEMBL4584288 0.74 TSHR (1.00) TSHRCHEK1METGSK3BLIMK1
SCHEMBL1450859 0.72 KMT2A (0.51) TSHRNPC1RAB9APOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012022776-A1 SUBSTITUTED THIOPENES OR FURANS AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2012-02-23 WO disclosed