SCHEMBL4584288

SCHEMBL4584288

O=C(O)c1csc(Br)c1Br

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 1.00
GPR35 Q9HC97 5/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
DAO P14920 1/20 0.35
GSK3B P49841 2/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
DAPK3 O43293 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
ABL1 P00519 1/20 0.35
NTRK1 P04629 1/20 0.35
RET P07949 1/20 0.35
MET P08581 1/20 0.35
PIM1 P11309 1/20 0.35
FGFR1 P11362 1/20 0.35
PDGFRA P16234 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28196417 0.79 TSHR (0.65) TSHRGPR35NPC1POLBGAA
SCHEMBL16212526 0.77 TSHR (0.63) TSHRGPR35NPC1POLBGAA
SCHEMBL18490191 0.77 TSHR (0.63) TSHRGPR35DAOGSK3BCHEK1
SCHEMBL673307 0.74 TSHR (0.59) TSHRNPC1POLBGAARAB9A
SCHEMBL2745234 0.73 NPC1 (0.59) TSHRGPR35NPC1POLBGAA
SCHEMBL9220569 0.71 TSHR (0.56) TSHRGPR35DAOGSK3BCES2
SCHEMBL12768622 0.71 TSHR (0.55) TSHRGPR35ALDH1A1ALOX15MAPT
SCHEMBL20607404 0.69 TSHR (0.52) TSHRGPR35DAOGSK3BCHEK1
SCHEMBL623033 0.68 TSHR (0.52) TSHRGPR35DAOGSK3BALAD
SCHEMBL852028 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed