SCHEMBL6739038

SCHEMBL6739038

CCOC(=O)N1CSC(C)(C)[C@@H]1C(=O)N[C@@H](Cc1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.56
ITGA4 P13612 20/20 0.56
ITGA2 P17301 1/20 0.56
ITGB7 P26010 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425741 0.94 ITGB1 (0.51) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6744281 0.91 ITGB1 (0.54) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6744929 0.85 ITGB1 (0.56) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6740614 0.85 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6745451 0.85 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6741663 0.85 ITGA4 (0.57) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6745542 0.85 ITGA4 (0.57) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6741753 0.80 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6745746 0.79 ITGB1 (0.58) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6742460 0.79 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
EP-1089989-A1 INHIBITORS OF ALPHA4BETA1 MEDIATED CELL ADHESION PHARMACIA & UPJOHN COMPANY (US) 2001-04-11 EP disclosed
WO-1999067230-A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION PHARMACIA & UPJOHN COMPANY (US) 1999-12-29 WO disclosed