SCHEMBL6739249

SCHEMBL6739249

COC(=O)[C@H](Cc1ccc(N(C(=O)c2c(Cl)cccc2Cl)C(=O)c2c(Cl)cccc2Cl)nc1)NC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.43
CTSL P07711 2/20 0.40
ITGB1 P05556 4/20 0.40
ITGA5 P08648 3/20 0.40
ITGB3 P05106 2/20 0.40
ITGAV P06756 1/20 0.40
CTSS P25774 5/20 0.39
CTSK P43235 4/20 0.39
CTSB P07858 2/20 0.38
ITGA4 P13612 2/20 0.38
ITGB7 P26010 2/20 0.38
ITGA2B P08514 1/20 0.38
EPHX2 P34913 1/20 0.37
NOS2 P35228 2/20 0.37
ACE P12821 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480191 0.82 KLK5 (0.43) KLK5CTSLITGB1ITGA5ITGB3
SCHEMBL7480195 0.82 KLK5 (0.43) KLK5CTSLITGB1ITGA5ITGB3
SCHEMBL763725 0.81 KLK5 (0.50) KLK5CTSLITGB3CTSSCTSK
Hydrochloric Acid SCHEMBL6740643 0.79 ITGB1 (0.40) ITGB1ITGA5ITGB3ITGAVITGA4
SCHEMBL28362228 0.77 ITGB3 (0.44) KLK5CTSLITGB3CTSSCTSK
SCHEMBL21896426 0.77 ITGB3 (0.44) KLK5CTSLITGB3CTSSCTSK
SCHEMBL6561292 0.77 ITGB1 (0.56) ITGB1ITGB3ITGAVITGA4ITGB7
SCHEMBL14799578 0.77 ITGB1 (0.56) ITGB1ITGB3ITGAVITGA4ITGB7
SCHEMBL12241473 0.77 KLK5 (0.50) KLK5CTSLITGB3CTSSCTSK
SCHEMBL33526968 0.77 KLK5 (0.50) KLK5CTSLITGB3CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed