SCHEMBL6740694

SCHEMBL6740694

COC(=O)[C@H](Cc1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1)NC(=O)C1CCCCN1C(=O)CCC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.50
ITGA4 P13612 19/20 0.50
ITGA2 P17301 1/20 0.46
ITGB7 P26010 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6739192 0.91 ITGA4 (0.55) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6743406 0.86 ITGB1 (0.50) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6743272 0.83 ITGA4 (0.54) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6740089 0.79 ITGA4 (0.51) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6740085 0.79 ITGA4 (0.51) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7423777 0.78 ITGB1 (0.51) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6742267 0.78 ITGA4 (0.54) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6739480 0.78 ITGA4 (0.54) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6739477 0.78 ITGA4 (0.54) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6745213 0.76 ITGA4 (0.55) ITGB1ITGA4ITGA2ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
EP-1089989-A1 INHIBITORS OF ALPHA4BETA1 MEDIATED CELL ADHESION PHARMACIA & UPJOHN COMPANY (US) 2001-04-11 EP disclosed
WO-1999067230-A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION PHARMACIA & UPJOHN COMPANY (US) 1999-12-29 WO disclosed