SCHEMBL6746352

SCHEMBL6746352

COP(=S)(Cl)OOC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744881 0.74 TSHR (0.37) TSHRTDP1
SCHEMBL1502255 0.71
Methylene Chloride SCHEMBL21985989 0.64
SCHEMBL5850459 0.64
SCHEMBL11793946 0.63 TSHR (0.37) TSHRTDP1
SCHEMBL6381874 0.61
SCHEMBL10604199 0.60
SCHEMBL11790662 0.58
SCHEMBL10882566 0.58
SCHEMBL11001130 0.58 TSHR (0.53) TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6699979-B2 PREPARED VIA A STEREOSPECIFIC SN2 NUCLEOPHILIC ATTACK OF A PHOSPHODIESTER, OR PHOSPHOROTHIOATE, ON THE 3' POSITION OF A XYLONUCLEOTIDE; USEFUL IN ANTISENSE OR PROBE TECHNOLOGY ISIS PHARMACEUTICALS, INC. 2004-03-02 US disclosed
US-6500945-B2 BIOSYNTHESIS; STEREOSPECIFIC ISIS PHARMACEUTICALS, INC. 2002-12-31 US disclosed
US-20020137921-A1 Oligonucleotides having chiral phosphorus linkages COOK PHILLIP DAN (US) 2002-09-26 US disclosed
EP-0655088-B1 OLIGONUCLEOTIDES HAVING CHIRAL PHOSPHORUS LINKAGES ISIS PHARMACEUTICALS INC (US) 2002-07-24 EP disclosed
US-20010008936-A1 Oligonucleotides having chiral phosphorus linkages ISIS PHARMACEUTICALS, INC. 2001-07-19 US disclosed
US-6239265-B1 FOR RESEARCH AND DIAGNOSIS ISIS PHARMACEUTICALS, INC. 2001-05-29 US disclosed
US-5852188-A Oligonucleotides having chiral phosphorus linkages ISIS PHARMACEUTICALS, INC. (US) 1998-12-22 US disclosed
US-5521302-A NUCLEOPHILIC REACTION OF PHOSPHATE GROUPS ISIS PHARMACEUTICALS, INC. (US) 1996-05-28 US disclosed
US-5212295-A Monomers for preparation of oligonucleotides having chiral phosphorus linkages ISIS PHARMACEUTICALS (US) 1993-05-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137921-A1 Oligonucleotides having chiral phosphorus linkages RNGTT, PNP, PSPH TSHR 1629/4885TDP1 582/4885
US-20010008936-A1 Oligonucleotides having chiral phosphorus linkages RNGTT, PNP, PSPH TSHR 1629/4885TDP1 582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.