SCHEMBL6747693

SCHEMBL6747693

N#Cc1nccnc1-c1ccc(CO)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
MAP2K4 P45985 2/20 0.38
CHEK1 O14757 1/20 0.37
PDE10A Q9Y233 2/20 0.36
RIPK1 Q13546 1/20 0.35
FYN P06241 1/20 0.35
BRAF P15056 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
EP300 Q09472 1/20 0.35
EGLN2 Q96KS0 1/20 0.34
ERBB2 P04626 4/20 0.33
S1PR1 P21453 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6749649 1.00 IKBKB (0.41) IKBKBCHUKMKNK1MKNK2MAP2K4
SCHEMBL6751316 0.83 ERBB2 (0.37) ERBB2
SCHEMBL11955055 0.83 CYP2A6 (0.46) PDE10AEP300ERBB2
SCHEMBL2475792 0.80 MMP3 (0.45) IKBKBCHUKERBB2
SCHEMBL985600 0.77 ERBB2 (0.56) CHEK1ERBB2
SCHEMBL29116345 0.77 ERBB2 (0.56) ERBB2CYP11B1CYP11B2
SCHEMBL14555800 0.77 ERBB2 (0.56) ERBB2
SCHEMBL10427642 0.76 ERBB2 (0.53) CHEK1ERBB2
SCHEMBL1521864 0.74 ERBB2 (0.35) CHEK1ERBB2
SCHEMBL8522790 0.73 MAP2K4 (0.47) MKNK1MKNK2MAP2K4PDE10ARIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058265-A1 COMPOUND LIBRARIES OF 2,3-SUBSTITUTED PYRAZINE DERIVATIVES CAPABLE OF BINDING TO G-PROTEIN COUPLED RECEPTORS BIOFOCUS PLC (GB) 2004-07-15 WO disclosed