SCHEMBL6747759

SCHEMBL6747759

NC(=O)c1nccnc1-c1ccc(C=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.40
PARP3 Q9Y6F1 1/20 0.40
ALDH1A1 P00352 4/20 0.36
ALDH5A1 P51649 1/20 0.35
ABAT P80404 1/20 0.35
KDM4E B2RXH2 3/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
DGAT1 O75907 1/20 0.32
IDO1 P14902 1/20 0.32
NEK2 P51955 1/20 0.32
PLK1 P53350 1/20 0.32
BRD4 O60885 1/20 0.32
ADORA2A P29274 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
CYP17A1 P05093 1/20 0.32
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28049210 0.79 NR3C2 (0.40) LMNAIDO1
SCHEMBL3468178 0.79 ADORA2A (0.50) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL28683096 0.78 PARP1 (0.45) PARP10PARP3ALDH1A1KDM4ELMNA
SCHEMBL30108240 0.78 PARP1 (0.45) PARP10PARP3ALDH1A1KDM4ELMNA
SCHEMBL6747763 0.75 MAPK1 (0.42) ALDH1A1ALDH5A1ABATKDM4ELMNA
SCHEMBL28982335 0.74 PTGS2 (0.49) LMNA
SCHEMBL8445737 0.72 BRD4 (0.46) ALDH1A1ALDH5A1ABATKDM4ELMNA
SCHEMBL30665107 0.70 MKNK1 (0.54) ALDH1A1LMNAMKNK1MKNK2CYP2A6
SCHEMBL30668220 0.70 MKNK1 (0.54) ALDH1A1LMNAMKNK1MKNK2CYP2A6
SCHEMBL2228105 0.70 MKNK1 (0.54) ALDH1A1LMNAMKNK1MKNK2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058265-A1 COMPOUND LIBRARIES OF 2,3-SUBSTITUTED PYRAZINE DERIVATIVES CAPABLE OF BINDING TO G-PROTEIN COUPLED RECEPTORS BIOFOCUS PLC (GB) 2004-07-15 WO disclosed