SCHEMBL6748010

SCHEMBL6748010

Cc1ccccc1CC(N)c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.45
ESR1 P03372 1/20 0.42
DPP4 P27487 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SOS2 Q07890 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
SCN4A P35499 5/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12706135 1.00 TAAR1 (0.45) TAAR1ESR1DPP4DPP7SLC6A2
SCHEMBL12706026 1.00 TAAR1 (0.45) TAAR1ESR1DPP4DPP7SLC6A2
SCHEMBL22295822 0.81 TAAR1 (0.37) TAAR1ESR1DPP4DPP7SLC6A2
SCHEMBL2339905 0.80 SCN4A (0.51) TAAR1SLC6A2SLC6A4SCN4A
SCHEMBL8410577 0.80 SCN4A (0.51) TAAR1SLC6A2SLC6A4SCN4A
SCHEMBL11323357 0.80 SLC6A2 (0.52) TAAR1ESR1SLC6A2SLC6A4CYP2D6
SCHEMBL9318564 0.79 ESR1 (0.45) TAAR1ESR1SLC6A2SLC6A4CYP3A4
SCHEMBL6547208 0.78 ESR1 (0.43) TAAR1ESR1SLC6A2SLC6A4CYP3A4
Ortetamine SCHEMBL42180 0.77 TAAR1 (0.52) TAAR1SLC6A2SLC6A4SOS2SLC6A3
SCHEMBL7591099 0.77 ESR1 (0.46) TAAR1ESR1SCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3690038-A1 ANTIBODY-PYRROLOBENZODIAZEPINE DERIVATIVE CONJUGATE DAIICHI SANKYO COMPANY, LIMITED (JP) 2020-08-05 EP disclosed
WO-2019065964-A1 ANTIBODY-PYRROLOBENZODIAZEPINE DERIVATIVE CONJUGATE 第一三共株式会社 2019-04-04 WO disclosed
US-9725405-B2 Alkynes and methods of reacting alkynes with 1,3-dipole-functional compounds UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2017-08-08 US disclosed
US-20040242437-A1 Antiwear performance of engine oils with $g(b)-dithiophosphorylated propionic acids CIBA SPECIALTY CHEMICALS CORP. 2004-12-02 US disclosed
WO-2002102945-A1 IMPROVED ANTIWEAR PERFORMANCE OF ENGINE OILS WITH $G(B)-DITHIOPHOSPHORYLATED PROPIONIC ACIDS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2002-12-27 WO disclosed
US-5892051-A WEAR RESISTANCE CIBA SPECIALTY CHEMICALS CORPORATION (US) 1999-04-06 US disclosed
US-5714442-A REACTING A 1H-1,2,4-TRIAZOLE OR BENZOTRIAZOLE WITH AN ALDEHYDE, OR DIOL OR DIVINYL ETHER; METAL DEACTIVATORS USED IN LUBRICANTS CIBA SPECIALITY CHEMICALS CORPORATION (US) 1998-02-03 US disclosed