SCHEMBL6748286

SCHEMBL6748286

CCCCOc1ccc(NC(=O)NC(c2ccc(C(=O)NCCC(=O)O)cc2)c2ccc(C3CCCCC3)cc2)cc1S(=O)(=O)CS(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.42
GCGR P47871 6/20 0.39
PPARD Q03181 2/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
EPHX2 P34913 2/20 0.37
GCG P01275 2/20 0.37
C5 P01031 1/20 0.35
ADCY6 O43306 3/20 0.35
ADCY3 O60266 3/20 0.35
ADCY9 O60503 3/20 0.35
ADCY5 O95622 3/20 0.35
ADCY8 P40145 3/20 0.35
ADCY7 P51828 3/20 0.35
ADCY2 Q08462 3/20 0.35
ADCY1 Q08828 3/20 0.35
ADCY4 Q8NFM4 3/20 0.35
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6751919 0.93 MCHR1 (0.44) MCHR1GCGRPPARDPPARGPPARA
SCHEMBL6751723 0.86 GCG (0.39) MCHR1GCGRGCGC5ADCY6
SCHEMBL6754063 0.85 GCGR (0.41) GCGRC5ADCY6ADCY3ADCY9
SCHEMBL6748283 0.84 GCGR (0.60) MCHR1GCGRADCY6ADCY3ADCY9
SCHEMBL6748285 0.83 GCGR (0.39) MCHR1GCGRPPARDPPARGPPARA
SCHEMBL6751922 0.81 EPHX2 (0.42) MCHR1GCGREPHX2GCG
SCHEMBL2651724 0.81 GCGR (0.49) MCHR1GCGRPPARDEPHX2ADCY6
SCHEMBL9071467 0.81 GCGR (0.51) MCHR1GCGRPPARDPPARGPPARA
SCHEMBL2659971 0.79 GCG (0.40) MCHR1GCGRGCGADCY6ADCY3
SCHEMBL6751739 0.78 GCGR (0.47) GCGRADCY6ADCY3ADCY9ADCY5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6706744-B2 HYPOGLYCEMIC AGENTS; ANTIDIABETIC AGENTS NOVO NORDISK A/S (DK) 2004-03-16 US claimed