SCHEMBL6749580

SCHEMBL6749580

COc1cccc(NCc2ccc(-c3nccnc3NS(=O)(=O)c3ccc(Cl)cc3)cc2)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 8/20 0.55
MAPT P10636 2/20 0.49
F2 P00734 1/20 0.46
DYRK1A Q13627 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
DYRK1B Q9Y463 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NAMPT P43490 1/20 0.46
TP53 P04637 1/20 0.46
GAA P10253 1/20 0.46
KDM1A O60341 1/20 0.44
MAOA P21397 1/20 0.44
ALOX12 P18054 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1964976 0.76 BCHE (0.63) MAPTDYRK1ACLK4DYRK1BALDH1A1
SCHEMBL2450795 0.76 PTGDR2 (0.66) PTGDR2
SCHEMBL6749573 0.75 PTGDR2 (0.65) PTGDR2
SCHEMBL2444500 0.71 PTGDR2 (1.00) PTGDR2
SCHEMBL10055018 0.70 NOS1 (0.63) MAPTALDH1A1LMNASMN1; SMN2GAA
SCHEMBL2446963 0.70 PTGDR2 (0.60) PTGDR2KDM1A
SCHEMBL2305041 0.70 MAPT (0.83) MAPTALDH1A1LMNAHPGDSMN1; SMN2
SCHEMBL6751910 0.69 PTGDR2 (0.57) PTGDR2ALDH1A1LMNASMN1; SMN2KDM1A
SCHEMBL2449413 0.68 PTGDR2 (0.57) PTGDR2ALDH1A1
SCHEMBL3132340 0.68 MAPT (0.87) MAPTALDH1A1LMNASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058265-A1 COMPOUND LIBRARIES OF 2,3-SUBSTITUTED PYRAZINE DERIVATIVES CAPABLE OF BINDING TO G-PROTEIN COUPLED RECEPTORS BIOFOCUS PLC (GB) 2004-07-15 WO disclosed