SCHEMBL6760168

SCHEMBL6760168

Cc1ncc(-c2cc(Cl)cc(NC(=O)c3cccc4c3[nH]c3ccc(F)cc34)c2)n1C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 11/20 0.41
GSK3B P49841 8/20 0.38
GRM5 P41594 1/20 0.38
MAPK1 P28482 2/20 0.37
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
IDO1 P14902 1/20 0.36
KAT5 Q92993 1/20 0.35
JAK2 O60674 1/20 0.35
CHRNA7 P36544 1/20 0.35
ICOSLG O75144 1/20 0.35
ICOS Q9Y6W8 1/20 0.35
KIT P10721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6760435 0.91 DYRK1A (0.45) DYRK1AGSK3BGRM5CLK2CLK3
SCHEMBL6804372 0.90 DYRK1A (0.45) DYRK1AGSK3BCLK2CLK3IDO1
SCHEMBL6755618 0.89 DYRK1A (0.40) DYRK1AGSK3BGRM5
SCHEMBL6756890 0.85 DYRK1A (0.44) DYRK1AGSK3BGRM5MAPK1CLK2
SCHEMBL6755637 0.81 MAPT (0.45) DYRK1AGSK3B
SCHEMBL6803727 0.80 DYRK1A (0.46) DYRK1AGSK3BGRM5CLK2CLK3
SCHEMBL6833169 0.73 DYRK1A (0.44) DYRK1AGSK3BGRM5CLK2CLK3
SCHEMBL6805348 0.72 DYRK1A (0.43) DYRK1AGSK3BGRM5CLK2CLK3
SCHEMBL6754360 0.72 DYRK1A (0.45) DYRK1AGSK3BGRM5MAPK1KAT5
SCHEMBL6832909 0.72 RAB9A (0.42) JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040087798-A1 Novel amide compounds FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-05-06 US disclosed
EP-1264820-A1 NOVEL AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-12-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087798-A1 Novel amide compounds H1-2, H1-0, H1-3 DYRK1A 3409/4885GSK3B 4671/4885GRM5 1930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.