SCHEMBL6760169

SCHEMBL6760169

COC(=O)CCSc1nccnc1SCCNC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
POLB P06746 1/20 0.40
IDO1 P14902 3/20 0.40
TDP1 Q9NUW8 2/20 0.39
HTT P42858 1/20 0.38
STK17B O94768 1/20 0.38
STK17A Q9UEE5 1/20 0.38
CYP3A4 P08684 1/20 0.38
TTK P33981 1/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
PTGS1 P23219 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
LMNA P02545 2/20 0.37
TSHR P16473 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MALT1 Q9UDY8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6762409 0.83 IDO1 (0.44) KDM4EPOLBIDO1TDP1HTT
SCHEMBL6757788 0.82 POLB (0.38) KDM4EPOLBIDO1STK17BSTK17A
SCHEMBL6762789 0.81 CYP3A4 (0.40) KDM4EIDO1TDP1HTTSTK17B
SCHEMBL5593747 0.78 TDP1 (0.46) KDM4EIDO1TDP1HTTCA12
SCHEMBL761060 0.78 KDM4E (0.42) KDM4EIDO1TDP1CYP3A4TTK
SCHEMBL1256643 0.74 TDP1 (0.55) KDM4ETDP1HTTCA12CA1
SCHEMBL10493769 0.73 IDO1 (0.46) IDO1TDP1HTTCYP3A4CA12
SCHEMBL28195039 0.73 IDO1 (0.41) IDO1TDP1HTTSTK17BSTK17A
Hydrochloric Acid SCHEMBL30168325 0.72 TDP1 (0.53) KDM4ETDP1HTTCA12CA1
SCHEMBL158052 0.72 SDCBP (0.61) IDO1TDP1CA1CA2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723716-B1 BACTERICIDE FOR STAPHYLOCOCCUS ESSENTIAL THERAPEUTICS, INC. 2004-04-20 US disclosed
EP-1222194-A1 7-ACYLAMINO-3-HETEROARYLTHIO-3-CEPHEM CARBOXYLIC ACID ANTIBIOTICS AND PRODRUGS THEREOF Essential Therapeutics, Inc. (US) 2002-07-17 EP disclosed
WO-2001021623-A1 7-ACYLAMINO-3-HETEROARYLTHIO-3-CEPHEM CARBOXYLIC ACID ANTIBIOTICS AND PRODRUGS THEREOF ESSENTIAL THERAPEUTICS, INC. (US) 2001-03-29 WO disclosed