SCHEMBL6764243

SCHEMBL6764243

CC(C)(C)Oc1ccc(C#N)c(C(F)(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AR P10275 20/20 0.63
PGR P06401 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13012268 0.83 AR (0.77) ARPGR
SCHEMBL22847930 0.80 MAOB (0.46) ARPGR
SCHEMBL4195488 0.80 AR (0.52) ARPGR
SCHEMBL20221049 0.79 AR (0.62) ARPGR
SCHEMBL13019733 0.79 TRPV4 (0.47) ARPGR
SCHEMBL4200970 0.79 AR (0.56) ARPGR
SCHEMBL13945827 0.79 AR (0.61) ARPGR
SCHEMBL4203274 0.79 AR (0.61) ARPGR
SCHEMBL13715641 0.79 AR (0.61) ARPGR
SCHEMBL4206006 0.79 AR (0.61) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183238-B2 Bicyclic and tricyclic compounds as KAT II inhibitors PFIZER INC. (US) 2012-05-22 US disclosed
US-20100324043-A1 Bicyclic And Tricyclic Compounds As KAT II Inhibitors PFIZER INC 2010-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324043-A1 Bicyclic And Tricyclic Compounds As KAT II Inhibitors KAT2A, KAT2B, KAT6B AR 2485/4885PGR 2907/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.