SCHEMBL6765739

SCHEMBL6765739

CC(C)(C)[Si](C)(C)Oc1ccc(O[Si](C)(C)C(C)(C)C)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.47
CA1 P00915 5/20 0.47
CA9 Q16790 5/20 0.47
PREP P48147 4/20 0.39
DRD2 P14416 1/20 0.35
ALDH1A1 P00352 4/20 0.33
MAPT P10636 3/20 0.33
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA14 Q9ULX7 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
PTPN1 P18031 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
ALOX12 P18054 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1828057 0.85 CA12 (0.47) CA12CA1CA9PREPDRD2
SCHEMBL15209708 0.85 CA12 (0.42) CA12CA1CA9PREPALDH1A1
SCHEMBL2090369 0.83 CA12 (0.49) CA12CA1CA9PREPHSP90AA1
SCHEMBL13478231 0.82 THRA (0.41) CA12CA1CA9CA2CA7
SCHEMBL2023774 0.82 CA12 (0.45) CA12CA1CA9PREPALDH1A1
SCHEMBL21409887 0.81 CYP1A2 (0.42) ALDH1A1MAPTMAPK1TDP1L3MBTL1
SCHEMBL6763269 0.81 CA12 (0.47) CA12CA1CA9PREPDRD2
SCHEMBL9013589 0.81 CA12 (0.47) CA12CA1CA9PREPDRD2
SCHEMBL23190575 0.80 CA12 (0.46) CA12CA1CA9PREPDRD2
SCHEMBL5517481 0.80 CA12 (0.46) CA12CA1CA9PREPPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130102740-A1 SULFONATED POLY(ARYLENE ETHER) COPOLYMER HAVING A CROSS-LINKABLE STRUCTURE, AND POLYELECTROLYTE MEMBRANE COMPRISING SAME GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2013-04-25 US disclosed
US-20130102740-A1 SULFONATED POLY(ARYLENE ETHER) COPOLYMER HAVING A CROSS-LINKABLE STRUCTURE, AND POLYELECTROLYTE MEMBRANE COMPRISING SAME GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2013-04-25 US disclosed
US-20130102740-A1 SULFONATED POLY(ARYLENE ETHER) COPOLYMER HAVING A CROSS-LINKABLE STRUCTURE, AND POLYELECTROLYTE MEMBRANE COMPRISING SAME GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2013-04-25 US disclosed
US-6726911-B1 SOLVENT EXTRACT; MICROBIOCIDES; ENDOPEPTIDASE, ANGIOTENSIN CONVERTING ENZYME AND SERUM-MEDIATED-BINDING OF LIPOPOLYSACCHARIDE INHIBITORS GANOMYCIN (DE) 2004-04-27 US disclosed
EP-1158995-B1 BIOLOGICALLY ACTIVE COMPOUNDS OF GANODERMA PFEIFFERI DMS 13239 GANOMYCIN GES FUER BIOMEDIZINI (DE) 2003-06-18 EP disclosed
EP-1158995-A1 BIOLOGICALLY ACTIVE COMPOUNDS OF GANODERMA PFEIFFERI DMS 13239 Ganomycin Gesellschaft für Biomedizinische Forschung mbH (DE) 2001-12-05 EP disclosed
WO-2000053207-A1 BIOLOGICALLY ACTIVE COMPOUNDS OF $I(GANODERMA PFEIFFERI) DMS 13239 GANOMYCIN GESELLSCHAFT FÜR BIOMEDIZINISCHE FORSCHUNG MBH ; (DE) 2000-09-14 WO disclosed