SCHEMBL6766495

SCHEMBL6766495

CC(=O)N(CCN1CCCC1)c1cc(C)[nH]c1/C=C1\C(=O)Nc2cccc(-c3cccc(F)c3)c21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 8/20 0.42
KDR P35968 7/20 0.42
FGFR1 P11362 4/20 0.42
TLK2 Q86UE8 1/20 0.42
KIT P10721 3/20 0.40
FLT3 P36888 5/20 0.40
ALK Q9UM73 3/20 0.40
FLT1 P17948 3/20 0.40
CSF1R P07333 2/20 0.40
PDGFRA P16234 1/20 0.40
CHEK1 O14757 1/20 0.39
ABL1 P00519 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
RET P07949 1/20 0.39
PHKG2 P15735 1/20 0.39
FGFR3 P22607 1/20 0.39
AXL P30530 1/20 0.39
ABL2 P42684 1/20 0.39
PTK2 Q05397 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6321236 0.81 PDGFRB (0.51) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6328657 0.79 PDGFRB (0.46) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6321318 0.78 FLT1 (0.45) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6322218 0.77 ALK (0.42) PDGFRBKDRFGFR1KITFLT3
SCHEMBL6319360 0.77 ALK (0.48) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6327898 0.77 KDR (0.38) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6765924 0.76 RET (0.62) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6324269 0.76 RET (0.62) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6329305 0.75 MET (0.43) PDGFRBKDRFGFR1TLK2KIT
SCHEMBL6323841 0.75 PDGFRB (0.57) PDGFRBKDRFGFR1TLK2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677368-B2 4-aryl substituted indolinones SUGEN, INC. 2004-01-13 US disclosed