SCHEMBL6768234

SCHEMBL6768234

COc1ccc2cnc(Nc3ccc(S(=O)(=O)c4ccccc4)cc3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.49
PDGFRB P09619 2/20 0.46
PDGFRA P16234 2/20 0.46
CDK1 P06493 2/20 0.46
KDR P35968 2/20 0.46
CDK2 P24941 1/20 0.46
TP53 P04637 2/20 0.46
MAPT P10636 2/20 0.46
PDE4B Q07343 3/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
PIK3CA P42336 1/20 0.45
NAMPT P43490 2/20 0.45
PLAU P00749 1/20 0.45
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1633099 0.86 IKBKB (0.65) IKBKBCDK1CDK2MAPTCA12
Hydrochloric Acid SCHEMBL28182076 0.85 PDGFRB (0.58) PDGFRBPDGFRACDK1KDRCDK2
SCHEMBL1633690 0.82 IKBKB (0.57) IKBKBCDK1CDK2CA12CA1
SCHEMBL1633112 0.81 BRD4 (0.56) IKBKBCDK1KDRCDK2MAPK1
SCHEMBL1634724 0.79 IKBKB (0.62) IKBKBCDK1CDK2CA12CA1
SCHEMBL1633172 0.78 KDM4E (0.59) IKBKBCDK2ALDH1A1HTTNPC1
SCHEMBL3320599 0.75 EGFR (0.76) PDGFRAKDRMAPTHTTNPC1
SCHEMBL1571219 0.73 IKBKB (0.48) IKBKBCDK1CDK2CA12CA1
SCHEMBL27780313 0.73 IKBKB (0.50) IKBKBCDK1KDRCDK2CA12
SCHEMBL8133819 0.73 BRAF (0.41) IKBKBPDGFRBCDK1KDRCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6727256-B1 4-AMINOQUINAZOLINE DERIVATIVES AS ANTICARCINOGENIC AGENTS SMITHKLINE BEECHAM CORPORATION 2004-04-27 US disclosed