SCHEMBL6770804

SCHEMBL6770804

Nc1nccc2cc(I)c(OCCNC(=O)OC(=O)C(F)(F)F)cc12

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 9/20 0.35
ROCK1 Q13464 4/20 0.35
F7 P08709 4/20 0.33
F3 P13726 1/20 0.33
KLK1 P06870 3/20 0.32
ATM Q13315 2/20 0.32
F9 P00740 1/20 0.32
F10 P00742 1/20 0.32
PLAU P00749 1/20 0.32
F11 P03951 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6770800 0.86 ROCK1 (0.38) KLKB1ROCK1F7F3KLK1
SCHEMBL6775414 0.85 ROCK1 (0.41) KLKB1ROCK1F7F3KLK1
SCHEMBL6770681 0.79 KLKB1 (0.32) KLKB1F7F9F10PLAU
Trifluoroacetic Acid SCHEMBL6770678 0.74 F7 (0.33) KLKB1ROCK1F7F9F10
SCHEMBL6771710 0.69 F10 (0.52) KLKB1F7KLK1F9F10
SCHEMBL6978093 0.68 F10 (0.40) F10PLAUPRSS1
SCHEMBL2544526 0.65 F12 (0.51) KLKB1ROCK1KLK1F9PLAU
SCHEMBL6776349 0.65 ROCK1 (0.46) ROCK1F10PLAU
SCHEMBL17787025 0.62 KLKB1 (0.42) KLKB1ROCK1KLK1ATMF9
SCHEMBL29728744 0.62 KLKB1 (0.42) KLKB1ROCK1KLK1ATMF9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825181-B1 ORALLY ADMINISTRATED TO EXHIBIT A STRONG ANTICOAGULANT EFFECT BY INHIBITING ACTIVATED BLOOD- COAGULATION FACTOR X AJINOMOTO CO., INC. (JP) 2004-11-30 US disclosed
EP-1065200-A1 AMINOISOQUINOLINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2001-01-03 EP disclosed