SCHEMBL6775414

SCHEMBL6775414

Nc1nccc2cc(I)c(OCCNC(=O)O)cc12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.41
F7 P08709 6/20 0.39
F3 P13726 3/20 0.39
ROCK2 O75116 1/20 0.36
KCNH2 Q12809 1/20 0.36
KLKB1 P03952 6/20 0.35
KLK1 P06870 5/20 0.35
F10 P00742 2/20 0.34
F11 P03951 2/20 0.34
F2 P00734 1/20 0.34
F9 P00740 1/20 0.34
PLAU P00749 1/20 0.34
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6770800 0.94 ROCK1 (0.38) ROCK1F7F3ROCK2KCNH2
SCHEMBL6770804 0.85 KLKB1 (0.35) ROCK1F7F3KLKB1KLK1
SCHEMBL6776349 0.79 ROCK1 (0.46) ROCK1F10PLAUALDH1A1
SCHEMBL6769241 0.76 ROCK1 (0.45) ROCK1PLAU
SCHEMBL6770030 0.75 ALDH1A1 (0.48) KLKB1PLAUKDM4EALDH1A1HPGD
Trifluoroacetic Acid SCHEMBL6770678 0.75 F7 (0.33) ROCK1F7KLKB1F10F11
SCHEMBL17786878 0.72 KLKB1 (0.46) KLKB1KLK1F10F9
SCHEMBL6770681 0.72 KLKB1 (0.32) F7KLKB1F10F11F9
SCHEMBL22733508 0.69 SMN1; SMN2 (0.42) KDM4EALDH1A1
SCHEMBL20781695 0.68 ROCK1 (0.64) ROCK1F7F3ROCK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825181-B1 ORALLY ADMINISTRATED TO EXHIBIT A STRONG ANTICOAGULANT EFFECT BY INHIBITING ACTIVATED BLOOD- COAGULATION FACTOR X AJINOMOTO CO., INC. (JP) 2004-11-30 US disclosed
EP-1065200-A1 AMINOISOQUINOLINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2001-01-03 EP disclosed