SCHEMBL6772813

SCHEMBL6772813

CCOC(=O)CCCn1c(NC(=O)c2cccs2)nc2cc(C(=O)NCC3CCCCC3)ccc21

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITK Q08881 18/20 0.69
TEC P42680 1/20 0.53
TXK P42681 1/20 0.53
INSR P06213 2/20 0.51
OPRK1 P41145 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6632540 0.88 ITK (0.72) ITKTECTXKINSROPRK1
SCHEMBL6766640 0.86 ITK (0.92) ITKTECTXK
SCHEMBL6770253 0.76 ITK (1.00) ITK
SCHEMBL6771407 0.76 ITK (0.88) ITKTECTXK
Hydrochloric Acid SCHEMBL8026086 0.75 CNR2 (0.49)
SCHEMBL8026960 0.75 CNR2 (0.51) ITK
SCHEMBL6770839 0.74 ITK (0.82) ITKTECTXK
SCHEMBL6771435 0.74 ITK (0.82) ITKTECTXK
SCHEMBL6632543 0.74 ITK (1.00) ITKTECTXK
SCHEMBL6771576 0.73 ITK (0.71) ITKINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825219-B2 NITROGEN COMPOUNDS SUCH AS 4-((5-(CYCLOHEXYL-METHYL-CARBAMOYL) -2(THIOPHENE-2-CARBONYL)-AMINO)BENZIMIDAZOL-1-YL)-BUTYRIC ACID ADMINISTERED FOR THE PROPHYLAXIS OF INFLAMMATORY, IMMUNOLOGICAL AND ALLERGIC DISORDERS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2004-11-30 US disclosed