SCHEMBL6776490

SCHEMBL6776490

COc1cc(OC)nc(OC(C(=O)O)C(C)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 20/20 0.76
EDNRA P25101 20/20 0.76
NR1I2 O75469 1/20 0.54
KCNE1 P15382 1/20 0.54
KCNQ1 P51787 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6781616 0.90 EDNRB (0.65) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL9369015 0.89 EDNRB (0.76) EDNRBEDNRANR1I2KCNE1KCNQ1
Darusentan SCHEMBL795084 0.85 EDNRB (1.00) EDNRBEDNRANR1I2KCNE1KCNQ1
Darusentan SCHEMBL1068546 0.85 EDNRB (1.00) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL8113638 0.84 EDNRB (0.77) EDNRBEDNRA
SCHEMBL4197434 0.83 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL4197423 0.83 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL8115354 0.83 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL6776058 0.83 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL12228356 0.83 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6686369-B1 α-hydrdroxylic acid derivatives, their production and use ABBOTT GMBH & CO., KG (DE) 2004-02-03 US disclosed