SCHEMBL6777360

SCHEMBL6777360

COc1cccc(-c2nn(-c3ccc(C(C)C)cc3)c3c2C(=O)C(C#N)C(C)(C)C3)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.39
DHODH Q02127 1/20 0.36
BTK Q06187 1/20 0.36
NAAA Q02083 3/20 0.35
NPBWR1 P48145 2/20 0.35
MCHR1 Q99705 2/20 0.35
SRC P12931 1/20 0.35
HPGD P15428 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 2/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6770531 0.87 MEN1 (0.40) OPRM1DHODHSRCHPGDALDH1A1
SCHEMBL6772794 0.87 CCNA2 (0.40) OPRM1DHODHBTKNAAANPBWR1
SCHEMBL6769818 0.87 OPRM1 (0.34) OPRM1DHODHNPBWR1MCHR1MEN1
SCHEMBL6771211 0.83 MEN1 (0.34) OPRM1DHODHSRCALDH1A1MEN1
SCHEMBL6770141 0.82 PTGS1 (0.41) OPRM1DHODHNPBWR1MCHR1HPGD
SCHEMBL7537240 0.81 OPRM1 (0.58) OPRM1DHODHSRCMAPT
SCHEMBL6770382 0.80 MEN1 (0.34) OPRM1NPBWR1MCHR1ALDH1A1GAA
SCHEMBL6767179 0.80 POLB (0.35) OPRM1DHODHHPGDALDH1A1GAA
SCHEMBL6766535 0.80 DHODH (0.36) OPRM1DHODHALDH1A1MEN1HTT
SCHEMBL6771166 0.79 OPRM1 (0.32) OPRM1NPBWR1MCHR1MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed