SCHEMBL6778472

SCHEMBL6778472

CCc1c(C(CC(=O)O)NC(=O)CNC(=O)c2cccc(NC(=N)N)c2)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.49
ITGAV P06756 14/20 0.49
ITGB6 P18564 12/20 0.49
ITGB1 P05556 4/20 0.49
ITGA5 P08648 4/20 0.49
ITGB5 P18084 4/20 0.49
ITGB8 P26012 4/20 0.49
ITGA8 P53708 4/20 0.49
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GPR139 Q6DWJ6 1/20 0.43
F7 P08709 1/20 0.41
EPHX2 P34913 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6777933 0.84 ITGB3 (0.64) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7835946 0.82 ITGB3 (0.51) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL6774023 0.82 ITGB3 (0.49) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL6783032 0.81 ITGB3 (0.72) ITGB3ITGAVITGB6ITGB1ITGA5
Trifluoroacetic Acid SCHEMBL3835291 0.80 ITGB3 (0.51) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL6776952 0.80 ITGB3 (0.49) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL242674 0.79 ITGB3 (0.55) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL6778768 0.78 ITGB3 (0.60) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7835684 0.78 ITGB3 (0.48) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL6776866 0.78 ITGB3 (0.53) ITGB3ITGAVITGB6ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831199-B1 In order to avoid bleeding side-effects when treating the conditions associated with integrin alpha v beta 3, it is beneficial to have compounds which are selective antagonists for alpha v beta 3 versus alpha IIb beta 3 G. D. SEARLE & CO. 2004-12-14 US disclosed