SCHEMBL6779947

SCHEMBL6779947

CC(C)CCn1cc(NC(=O)c2ccc3[nH]c(C(=O)Nc4cc(C(=O)Nc5cc(C(=O)NCCCN(C)C)n(C)c5)n(CCC(C)C)c4)cc3c2)cc1C(=O)Nc1cc(C(=O)NCCCN(C)C)n(C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRAS P01112 4/20 0.52
ESR1 P03372 4/20 0.52
ESR2 Q92731 4/20 0.52
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
PRKCA P17252 3/20 0.43
ITGB3 P05106 2/20 0.40
ITGA2B P08514 2/20 0.40
HRH4 Q9H3N8 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NR4A1 P22736 1/20 0.39
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1843199 0.87 HRAS (0.47) HRASESR1ESR2HDAC1HDAC2
SCHEMBL5889539 0.85 HRAS (0.60) HRASESR1ESR2HDAC1HDAC2
SCHEMBL5889621 0.84 HRAS (0.54) HRASESR1ESR2ITGB3ITGA2B
SCHEMBL5889846 0.83 HRAS (0.54) HRASESR1ESR2ITGB3ITGA2B
SCHEMBL1842501 0.82 HDAC1 (0.48) HRASESR1ESR2HDAC1HDAC2
SCHEMBL3563935 0.82 HRAS (0.43) HRASESR1ESR2HDAC1HDAC2
SCHEMBL1843141 0.81 SIGMAR1 (0.47) HDAC1HDAC2HDAC8PRKCAKDM4E
SCHEMBL5677699 0.80 HRAS (0.50) HRASESR1ESR2ITGB3ITGA2B
SCHEMBL1842079 0.80 HRAS (0.55) HRASESR1ESR2HDAC1HDAC2
SCHEMBL5896881 0.79 HRAS (0.51) HRASESR1ESR2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1467969-A2 DNA MINOR GROOVE BINDING COMPOUNDS The University of Strathclyde (GB) 2004-10-20 EP claimed
WO-2003059881-A2 DNA MINOR GROOVE BINDING COMPOUNDS UNIVERSITY OF STRATHCLYDE (GB) 2003-07-24 WO claimed