SCHEMBL6783287

SCHEMBL6783287

CCCCNCCCCC(=O)Nc1cccc(-c2n[nH]c(=O)c3ccccc23)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.55
ROCK2 O75116 2/20 0.49
ROCK1 Q13464 2/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
HPGD P15428 2/20 0.48
USP2 O75604 1/20 0.48
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 3/20 0.46
LMNA P02545 2/20 0.46
AURKA O14965 1/20 0.45
PDE5A O76074 1/20 0.45
PDE1A P54750 1/20 0.45
PDE1B Q01064 1/20 0.45
PDE3B Q13370 1/20 0.45
PDE1C Q14123 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6788534 0.99 PARP1 (0.54) PARP1ROCK2ROCK1SMN1; SMN2HPGD
SCHEMBL6782921 0.96 PARP1 (0.55) PARP1ROCK2ROCK1SMN1; SMN2HPGD
Hydrochloric Acid SCHEMBL6788444 0.95 PARP1 (0.54) PARP1ROCK2ROCK1SMN1; SMN2HPGD
SCHEMBL6792847 0.93 PARP1 (0.53) PARP1ROCK2ROCK1SMN1; SMN2HPGD
SCHEMBL6782566 0.93 PARP1 (0.60) PARP1ROCK2ROCK1SMN1; SMN2HPGD
SCHEMBL6793941 0.92 PARP1 (0.61) PARP1ROCK2ROCK1SMN1; SMN2HPGD
SCHEMBL6788872 0.91 ROCK1 (0.50) PARP1ROCK2ROCK1HPGDNPSR1
SCHEMBL6782927 0.90 PARP1 (0.48) PARP1ROCK2ROCK1KDM4EALDH1A1
SCHEMBL6782343 0.90 ROCK1 (0.49) PARP1ROCK2ROCK1HPGDNPSR1
Hydrochloric Acid SCHEMBL6794797 0.90 ROCK1 (0.49) PARP1ROCK2ROCK1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677333-B1 ANTIISCHEMIC AGENTS; BRAIN, CARDIOVASCULAR, MUSCULAR, AND GASTROINTESTINAL DISORDERS; ANALGESICS, ANTIDIABETIC AGENTS; RETROVIRUS SENSITIZERS; ALZHEIMER*S DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2004-01-13 US claimed
EP-1148053-A1 2H-PHTHALAZIN-1-ONE DERIVATIVES AND DRUGS COMPRISING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-24 EP claimed