SCHEMBL6788872

SCHEMBL6788872

O=C(CCCCNCCO)Nc1cccc(-c2n[nH]c(=O)c3ccccc23)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.50
ROCK2 O75116 3/20 0.50
PARP1 P09874 4/20 0.48
HPGD P15428 2/20 0.46
HDAC6 Q9UBN7 4/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
AURKA O14965 2/20 0.43
AURKB Q96GD4 1/20 0.43
MAP2K7 O14733 1/20 0.43
ATM Q13315 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6794797 0.99 ROCK1 (0.49) ROCK1ROCK2PARP1HPGDHDAC6
SCHEMBL6782921 0.91 PARP1 (0.55) ROCK1ROCK2PARP1HPGDHDAC6
SCHEMBL6782343 0.91 ROCK1 (0.49) ROCK1ROCK2PARP1HPGDHDAC6
SCHEMBL6783287 0.91 PARP1 (0.55) ROCK1ROCK2PARP1HPGDHDAC6
SCHEMBL6782474 0.91 ROCK1 (0.55) ROCK1ROCK2PARP1HPGDHDAC6
Hydrochloric Acid SCHEMBL6788444 0.90 PARP1 (0.54) ROCK1ROCK2PARP1HPGDHDAC6
Hydrochloric Acid SCHEMBL6788557 0.90 ROCK1 (0.48) ROCK1ROCK2PARP1HPGDHDAC6
Hydrochloric Acid SCHEMBL6788534 0.90 PARP1 (0.54) ROCK1ROCK2PARP1HPGDHDAC6
SCHEMBL6792847 0.90 PARP1 (0.53) ROCK1ROCK2PARP1HPGDHDAC6
SCHEMBL6782927 0.89 PARP1 (0.48) ROCK1ROCK2PARP1HDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677333-B1 ANTIISCHEMIC AGENTS; BRAIN, CARDIOVASCULAR, MUSCULAR, AND GASTROINTESTINAL DISORDERS; ANALGESICS, ANTIDIABETIC AGENTS; RETROVIRUS SENSITIZERS; ALZHEIMER*S DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2004-01-13 US claimed
EP-1148053-A1 2H-PHTHALAZIN-1-ONE DERIVATIVES AND DRUGS COMPRISING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-24 EP claimed