SCHEMBL6784008

SCHEMBL6784008

Cc1cc(C)c(-n2cc(C)c3c(=O)[nH]c(C)nc32)c(C)c1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 12/20 0.55
CCND1 P24385 12/20 0.55
PARP1 P09874 2/20 0.45
FPR3 P25089 2/20 0.43
TSPO P30536 2/20 0.43
CRHR1 P34998 2/20 0.43
TMEM97 Q5BJF2 2/20 0.43
CCNE2 O96020 2/20 0.39
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6218669 0.82 CDK4 (0.42) CDK4CCND1PARP1CCNE2CCNE1
SCHEMBL6217714 0.82 CDK4 (0.41) CDK4CCND1PARP1CCNE2CCNE1
SCHEMBL6218693 0.77 CDK4 (0.46) CDK4CCND1PARP1CCNE2CCNE1
SCHEMBL6213926 0.77 CDK4 (0.47) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL4562079 0.77 CA12 (0.49) CDK4CCND1PARP1CCNE1CDK2
SCHEMBL6780074 0.75 CDK4 (0.57) CDK4CCND1PARP1CRHR1CCNE2
SCHEMBL6218319 0.75 CDK4 (0.36) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL6213942 0.75 CDK4 (0.43) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL6216498 0.74 PDE2A (0.39) CDK4CCND1CRHR1CA12CA1
SCHEMBL6216009 0.72 CDK4 (0.36) CDK4CCND1CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6765008-B1 PYRROLO(2,3-D)PYRIMIDINE DERIVATIVES; ANXIOLYTIC AGENTS; NERVOUS SYSTEM, BRAIN, PSYCHOLOGICAL, EATING, AND GASTROINTESTINAL DISORDERS; CORTICOTROPIN-RELEASING FACTOR ANTAGONISTS PFIZER INC 2004-07-20 US disclosed
EP-0674641-B1 PYRROLOPYRIMIDINES AS CRF ANTAGONISTS PFIZER (US) 1999-03-03 EP disclosed
WO-1994013676-A1 PYRROLOPYRIMIDINES AS CRF ANTAGONISTS PFIZER INC. (US) 1994-06-23 WO disclosed