SCHEMBL678486

SCHEMBL678486

COc1c(O)c(C(C)=O)c(OC)c(OC)c1OC

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 2/20 0.53
CYP3A4 P08684 3/20 0.44
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.40
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KCNA2 P16389 1/20 0.38
KCNA4 P22459 1/20 0.38
KCNA5 P22460 1/20 0.38
KCNA1 Q09470 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25383713 0.85 PTPN1 (0.50) KCNA3CYP3A4KCNA2KCNA4KCNA5
SCHEMBL11106706 0.84 CYP3A4 (0.48) KCNA3CYP3A4MEN1HPGDKMT2A
SCHEMBL684711 0.84 KCNA3 (0.49) KCNA3CYP3A4
SCHEMBL4108349 0.83 KCNA3 (0.47) KCNA3CYP3A4LMNAUSP2MAPK1
SCHEMBL5589033 0.83 KDM4E (0.45) KCNA3CYP3A4MEN1HPGDKMT2A
SCHEMBL25384697 0.82 PTPN1 (0.52) KCNA3CYP3A4LMNAUSP2MAPK1
Potassium Ion SCHEMBL29141174 0.79 KCNA3 (0.38) KCNA3CYP3A4LMNASMN1; SMN2
SCHEMBL9752628 0.78 CYP3A4 (0.52) KCNA3CYP3A4MEN1HPGDKMT2A
SCHEMBL25952524 0.78 CYP3A4 (0.52) KCNA3CYP3A4MEN1HPGDKMT2A
SCHEMBL25952538 0.78 CYP3A4 (0.52) KCNA3CYP3A4MEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110287106-A1 COGNITIVE IMPAIRMENT AMELIORANT JAPAN ROYAL JELLEY CO., LTD. (JP) 2011-11-24 US claimed
EP-2311472-A1 COGNITIVE DISORDER-AMELIORATING AGENT Japan Royal Jelly Co., Ltd. (JP) 2011-04-20 EP claimed
US-11559512-B2 Composition for prevention, alleviation, and/or treatment of heat illness TOYO UNIVERSITY (JP) 2023-01-24 US disclosed
CN-110498784-B Nobiletin derivatives or pharmaceutically acceptable salts thereof, and preparation method and application thereof 广东克冠达医药科技有限公司 2022-06-14 CN disclosed
US-20200297694-A1 COMPOSITION FOR PREVENTION, ALLEVIATION, AND/OR TREATMENT OF HEAT ILLNESS TOYO UNIVERSITY (JP) 2020-09-24 US disclosed
EP-3689345-A1 COMPOSITION FOR PREVENTION, ALLEVIATION, AND/OR TREATMENT OF HEAT STROKE Toyo University (JP) 2020-08-05 EP disclosed
EP-2311472-B1 COGNITIVE DISORDER-AMELIORATING AGENT JAPAN ROYAL JELLY CO LTD (JP) 2014-03-05 EP disclosed
EP-2311472-B1 COGNITIVE DISORDER-AMELIORATING AGENT JAPAN ROYAL JELLY CO LTD (JP) 2014-03-05 EP disclosed
US-20130129832-A1 COGNITIVE IMPAIRMENT AMELIORANT TOHOKU UNIVERSITY (JP) 2013-05-23 US disclosed
US-20130129832-A1 COGNITIVE IMPAIRMENT AMELIORANT TOHOKU UNIVERSITY (JP) 2013-05-23 US disclosed
US-20110287106-A1 COGNITIVE IMPAIRMENT AMELIORANT JAPAN ROYAL JELLEY CO., LTD. (JP) 2011-11-24 US disclosed
US-20110287106-A1 COGNITIVE IMPAIRMENT AMELIORANT JAPAN ROYAL JELLEY CO., LTD. (JP) 2011-11-24 US disclosed
EP-2311472-A1 COGNITIVE DISORDER-AMELIORATING AGENT Japan Royal Jelly Co., Ltd. (JP) 2011-04-20 EP disclosed
EP-2311472-A1 COGNITIVE DISORDER-AMELIORATING AGENT Japan Royal Jelly Co., Ltd. (JP) 2011-04-20 EP disclosed
US-4532254-A Inhibitor of aldose reductase KAKEN PHARMACEUTICAL CO., LTD. (JP) 1985-07-30 US disclosed
EP-0118571-A1 Inhibitor of aldose reductase Kaken Pharmaceutical Co., Ltd. (JP) 1984-09-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11559512-B2 Composition for prevention, alleviation, and/or treatment of heat illness TNF, HSF1, HSP90AA1 KCNA3 2497/4885CYP3A4 1707/4885MEN1 3508/4885
US-20130129832-A1 COGNITIVE IMPAIRMENT AMELIORANT CHAT, ACHE, PSEN1 KCNA3 4482/4885CYP3A4 4098/4885MEN1 3488/4885
US-20200297694-A1 COMPOSITION FOR PREVENTION, ALLEVIATION, AND/OR TREATMENT OF HEAT ILLNESS TNF, HSF1, HSP90AA1 KCNA3 2497/4885CYP3A4 1707/4885MEN1 3508/4885
US-20110287106-A1 COGNITIVE IMPAIRMENT AMELIORANT CHAT, ACHE, PSEN1 KCNA3 4482/4885CYP3A4 4098/4885MEN1 3488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.