SCHEMBL6788006

SCHEMBL6788006

O=C(CI)c1ccc(Br)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 1.00
HDAC1 Q13547 3/20 0.59
HDAC8 Q9BY41 3/20 0.59
HDAC3 O15379 1/20 0.59
HDAC4 P56524 1/20 0.59
HDAC7 Q8WUI4 1/20 0.59
HDAC2 Q92769 1/20 0.59
HDAC10 Q969S8 1/20 0.59
HDAC11 Q96DB2 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
HDAC9 Q9UKV0 1/20 0.59
HDAC5 Q9UQL6 1/20 0.59
OGG1 O15527 1/20 0.56
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
HAO1 Q9UJM8 1/20 0.50
NPC1 O15118 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10020269 0.87 GSK3B (0.76) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL3469826 0.83 GSK3B (0.71) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL241664 0.80 GSK3B (0.70) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL1305020 0.80 GSK3B (0.70) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL12139286 0.79 GSK3B (0.64) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL28443057 0.78 GSK3B (0.64) GSK3BCA1CA2NPC1HPGD
SCHEMBL70930 0.78 GSK3B (1.00) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL55916 0.78 GSK3B (0.67) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL11695106 0.78 GSK3B (0.64) GSK3BCA1CA2NPC1RAB9A
SCHEMBL658726 0.76 GSK3B (0.64) GSK3BCES2CES1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685458-B Organic compound and application thereof 广州华睿光电材料有限公司 2024-03-08 CN disclosed
CN-114685454-B Organic compounds, mixtures, compositions and organic electronic devices 广州华睿光电材料有限公司 2024-01-12 CN disclosed
WO-2023115621-A1 METHOD FOR PREPARING Α-HALOGENATED ACETOPHENONE COMPOUND UNDER CATALYSIS OF IONIC LIQUID [TEA][TFOH]2 大连大学 2023-06-29 WO disclosed
CN-114685454-A Organic compound, mixture, composition and organic electronic device 广州华睿光电材料有限公司 2022-07-01 CN disclosed
CN-114685458-A Organic compound and application thereof 广州华睿光电材料有限公司 2022-07-01 CN disclosed
WO-2015005901-A1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-01-15 WO disclosed
WO-2013106520-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2013-07-18 WO disclosed
US-20070296101-A1 cross-linked polyaryletherketone polymers are used as the recording layers in atomic force data storage devices, giving significantly improved performance when compared to previously reported cross-linked and linear polymers INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2007-12-27 US disclosed
WO-2007120454-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM LLC (BM) 2007-10-25 WO disclosed
US-6747057-B2 SUCH 1-(2-BROMO-4,5-DICHLORO-THIOPHEN-3-YL)-2-CHLORO-ETHANONE FOR TREATMENT OF ALZHEIMER'S DISEASE OR DIABETES CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS (ES) 2004-06-08 US disclosed
US-20030199508-A1 Compounds and their therapeutic use UNIVERSIDAD AUTONOMA DE MADRID (UAM) (ES) 2003-10-23 US disclosed
WO-2003055479-A1 COMPOUNDS AND THEIR THERAPEUTIC USE RELATED TO THE PHOSPHORYLATING ACTIVITY OF THE ENZYME GSK-3 CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS (ES) 2003-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030199508-A1 Compounds and their therapeutic use CNKSR1, CBR1, CBR3 GSK3B 4/4885HDAC1 621/4885HDAC8 1036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.