SCHEMBL6792275

SCHEMBL6792275

C/C(=C/C(=O)Nc1ccc(F)cc1C(=O)O)c1ccc(Cl)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.53
PPARA Q07869 1/20 0.53
KDM4E B2RXH2 1/20 0.52
HSD17B10 Q99714 1/20 0.52
TSHR P16473 1/20 0.47
CASP1 P29466 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GRIK1 P39086 2/20 0.45
DHODH Q02127 3/20 0.44
AVPR2 P30518 1/20 0.44
OXTR P30559 1/20 0.44
AVPR1A P37288 1/20 0.44
TERT O14746 3/20 0.43
TP53 P04637 1/20 0.43
FABP3 P05413 1/20 0.42
FABP4 P15090 1/20 0.42
SERPINE1 P05121 1/20 0.42
PYGL P06737 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6785956 0.82 TERT (0.53) KDM4EHSD17B10TSHRDHODHTERT
SCHEMBL6784709 0.81 TERT (0.46) PPARGPPARAKDM4EHSD17B10DHODH
SCHEMBL6787442 0.80 MAPT (0.56) PPARGPPARAKDM4EHSD17B10TSHR
SCHEMBL6790635 0.77 TERT (0.52) DHODHTERT
SCHEMBL6785267 0.77 KDM4E (0.57) PPARGPPARAKDM4EHSD17B10TERT
SCHEMBL6782589 0.77 DHODH (0.58) KDM4EDHODHTERTFABP3FABP4
SCHEMBL6785899 0.76 TERT (0.54) KDM4EDHODHAVPR2OXTRAVPR1A
SCHEMBL6787380 0.74 MEN1 (0.52) TSHRGRIK1DHODHTERT
SCHEMBL4020296 0.74 TERT (0.77) KDM4EDHODHTERT
SCHEMBL6784596 0.74 DHODH (0.48) DHODHTERTFABP3FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6727250-B2 ADMINISTERING COMPOUNDS SUCH AS TRANS-3-(NAPHTH-2-YL)-BUT-2-ENOIC ACID-N-(2-CARBOXY-PHENYL)-AMIDE OR LIKE FOR THERAPY OF CONDITIONS ASSOCIATED WITH INCREASED TELOMERASE ACTIVITY, E.G. TUMOUR DISEASES BOEHRINGER INGELHEIM PHARMA KG (DE) 2004-04-27 US claimed
US-6727250-B2 ADMINISTERING COMPOUNDS SUCH AS TRANS-3-(NAPHTH-2-YL)-BUT-2-ENOIC ACID-N-(2-CARBOXY-PHENYL)-AMIDE OR LIKE FOR THERAPY OF CONDITIONS ASSOCIATED WITH INCREASED TELOMERASE ACTIVITY, E.G. TUMOUR DISEASES BOEHRINGER INGELHEIM PHARMA KG (DE) 2004-04-27 US disclosed
US-20020099089-A1 Carboxylic acid amides, pharmaceutical compositions containing these compounds, their use and preparation BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2002-07-25 US disclosed
US-6362210-B1 ANTITUMOR, ANTICANCER AGENT BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020099089-A1 Carboxylic acid amides, pharmaceutical compositions containing these compounds, their use and preparation TERT, NAT1, POT1 PPARG 151/4885PPARA 86/4885KDM4E 1243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.