SCHEMBL6793396

SCHEMBL6793396

CN1CCN(CCCn2nc3c(c2C(=O)O)CCc2cnccc2-3)CC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.36
GSK3B P49841 1/20 0.34
IKBKE Q14164 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
CHRM1 P11229 1/20 0.32
RAB9A P51151 1/20 0.32
AURKA O14965 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6787046 0.93 CDK2 (0.38) NAMPTCHRM1AURKACCNA2CDK2
SCHEMBL6793766 0.92 CCNA2 (0.39) NAMPTAURKACCNA2CDK2CCNA1
SCHEMBL6794733 0.91 BRAF (0.34) NAMPTGSK3B
SCHEMBL1659385 0.86 CDK2 (0.34) NAMPTAURKACCNA2CDK2CCNA1
Trifluoroacetic Acid SCHEMBL6796768 0.85 CCNC (0.32) ALDH1A1CHRM1AURKACCNA2CDK2
SCHEMBL6793304 0.85 KDM4C (0.37) AURKACCNA2CDK2CCNA1
Hydrochloric Acid SCHEMBL1658167 0.84 CDK2 (0.42) AURKACCNA2CDK2CCNA1
SCHEMBL6793189 0.84 CDK2 (0.35) AURKACCNA2CDK2CCNA1
Trifluoroacetic Acid SCHEMBL6791881 0.84 CHRM2 (0.35) CHRM1AURKACCNA2CDK2CCNA1
Hydrochloric Acid SCHEMBL4263501 0.84 CYP3A4 (0.34) NAMPTCHRM1AURKACCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040127492-A1 Cyclic pyrazoles for the inhibition of mitogen activated protein kinase-activated protein kinase-2 PHARMACIA CORPORATION 2004-07-01 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127492-A1 Cyclic pyrazoles for the inhibition of mitogen activated protein kinase-activated protein kinase-2 MKNK2, MAPKAPK2, MAP3K2 NAMPT 658/4885GSK3B 447/4885IKBKE 511/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.