SCHEMBL6796908

SCHEMBL6796908

F[C@H]1CCC[C@@H]1Nc1nc2cncnc2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.34
LATS1 O95835 2/20 0.32
LATS2 Q9NRM7 1/20 0.32
HCRTR1 O43613 1/20 0.31
BRD4 O60885 1/20 0.31
PIM1 P11309 3/20 0.31
JAK3 P52333 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6796013 1.00 IRAK4 (0.34) IRAK4LATS1LATS2HCRTR1BRD4
SCHEMBL7662481 0.79 RIPK1 (0.46) IRAK4LATS1LATS2PIM1
SCHEMBL6797408 0.73 PIM1 (0.43) IRAK4BRD4PIM1
Hydrochloric Acid SCHEMBL9602450 0.72 PIM1 (0.43) IRAK4BRD4PIM1
Bromide SCHEMBL9602726 0.72 PIM1 (0.43) IRAK4BRD4PIM1
Water SCHEMBL9602231 0.72 PIM1 (0.43) IRAK4BRD4PIM1
Hydrochloric Acid SCHEMBL9688940 0.72 PIM1 (0.48) BRD4PIM1
Bromide SCHEMBL9602934 0.72 RPS6KB1 (0.33)
SCHEMBL3952312 0.69 KDM4E (0.40)
SCHEMBL9654498 0.68 EGFR (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677316-B2 TREATING ISCHEMIA, CARDIOVASCULAR DISORDERS, STROKE, PAIN, NERVOUS SYSTEM DISORDERS OR SLEEP APNEA; ADENOSINE A1 RECEPTOR AGONIST; 2-(3-(TERT-BUTYL)-1,2,4-OXADIAZOL-5-YL)-5-(6-(ISOBUTYLAMINO)-9H-PURIN-9-YL) TETRAHYDROFURAN-3,4-DIOL SMITHKLINE BEECHAM CORPORATION 2004-01-13 US disclosed