SCHEMBL6798778

SCHEMBL6798778

CC1(C)OB(c2cccc(-n3cnc4cc(-c5ccoc5)cnc43)c2)OC1(C)C

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.45
LPL P06858 2/20 0.44
LIPG Q9Y5X9 2/20 0.44
GAK O14976 2/20 0.41
KDR P35968 1/20 0.34
HPGD P15428 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
CHRNA7 P36544 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804619 0.79 NT5E (0.69) NT5EGAKKDRHPGD
SCHEMBL6799283 0.77 NT5E (0.47) NT5EGAKKDRKCNH2
SCHEMBL6797821 0.75 NT5E (0.47) NT5EGAKKDR
SCHEMBL7417006 0.73 NT5E (0.45) NT5EGAKKDRHPGD
SCHEMBL6796978 0.72 NT5E (0.45) NT5EGAKKDRHPGD
SCHEMBL6804409 0.71 NT5E (0.44) NT5EGAKKDRHPGD
SCHEMBL6807826 0.71 NT5E (0.44) NT5EGAKKDRHPGD
SCHEMBL6803894 0.71 NT5E (0.44) NT5EGAKKDRHPGD
SCHEMBL6799281 0.71 NT5E (0.43) NT5EGAKKDRHPGD
SCHEMBL6803865 0.69 NT5E (0.42) NT5EGAKKDRHPGDIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723735-B1 TREATMENT OR PREVENTION OF ANXIETY MERCK SHARP & DOHME LTD. 2004-04-20 US disclosed
EP-1214319-B1 IMIDAZO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2003-11-26 EP disclosed